Details of the Active Pharmaceutical Ingredient (API)
General Information of API (ID: D00296) | |||||
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Name |
Gabapentin
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Synonyms |
Click to Show/Hide the Synonyms of This API
gabapentin; 60142-96-3; Neurontin; 1-(Aminomethyl)cyclohexaneacetic acid; Gabapentine; Aclonium; 2-[1-(aminomethyl)cyclohexyl]acetic acid; Gabapetin; Gabapentinum; Fanatrex; Gabapentino; Gabapen; Serada; [1-(AMINOMETHYL)CYCLOHEXYL]ACETIC ACID; Cyclohexaneacetic acid, 1-(aminomethyl)-; 2-(1-(aminomethyl)cyclohexyl)acetic acid; gabapentina; Gralise; (1-Aminomethyl-cyclohexyl)-acetic acid; Go 3450; Goe-3450; GOE 2450; CI 945; CI-945; C9H17NO2; DM-1796; GOE 3450; UNII-6CW7F3G59X; Gabarone; 1-(Aminomethyl)-cyclohexaneacetic acid; Gabapentin free base; DM-5689; MFCD00865286; CHEMBL940; GABAPENTIN; NEURONTIN; 6CW7F3G59X; CHEBI:42797; 60142-96-3 (free base); Gabapentino [Spanish]; Gabapentine [INN-French]; Gabapentinum [INN-Latin]; NCGC00015466-08; DSSTox_CID_74; Gabapentino [INN-Spanish]; Vultin; CAS-60142-96-3; Gabapentin GR; DSSTox_RID_75350; DSSTox_GSID_20074; gabapentinium; gabapentin (Neurontin); Neuontin; Sefelsa; Therapentin-90; Neurontin (TN); CCRIS 7210; HSDB 7364; SR-01000000019; EINECS 262-076-3; BRN 2359739; Neurentin; Gabapentin-ER; Novo-Gabapentine; Gabapentin, solid; Gabapentin [USAN:USP:INN:BAN]; Gabapentin solution; DDS-2003; Prestwick_151; 1-(Aminomethyl)cyclohexaneaceticAcid; Gralise (TN); Neurontin,Gabapentin; GABAPETINE; Tocris-0806; Lopac-G-154; Prestwick0_000861; Prestwick1_000861; Prestwick2_000861; Prestwick3_000861; SCHEMBL8343; Lopac0_000582; BSPBio_000901; Gabapentin (JAN/USP/INN); MLS000069358; BIDD:GT0656; SPBio_002822; BPBio1_000993; GTPL5483; ZINC4949; DTXSID0020074; HMS1570N03; HMS2089J03; HMS2097N03; HMS2236O03; HMS3261F06; HMS3650A20; HMS3714N03; 1-aminomethyl cyclohexaneacetic acid; 1-aminomethylcyclohexane acetic acid; ACT03340; BCP25698; HY-A0057; 1-(aminomethyl)cyclohexanacetic acid; Tox21_110157; Tox21_500582; ANW-43124; BBL010794; BDBM50080153; NSC742194; SBB066157; STK598009; 1-(aminomethyl)cyclohexyl-acetic Acid; 1-amino methyl cyclohexane-acetic acid; AKOS000280865; Tox21_110157_1; 1-Aminomethyl-1cyclohexane-acetic acid; 2-[(aminomethyl)cyclohexyl]acetic acid; AB07485; AC-1485; CCG-204671; CS-1545; DB00996; KS-1064; LP00582; MCULE-5392848565; NSC-742194; SDCCGSBI-0050564.P002; 1-aminomethyl-1-cyclohexane-acetic acid; NCGC00015466-01; NCGC00015466-02; NCGC00015466-03; NCGC00015466-04; NCGC00015466-05; NCGC00015466-06; NCGC00015466-07; NCGC00015466-09; NCGC00015466-11; NCGC00015466-27; NCGC00016891-01; NCGC00021545-02; NCGC00021545-04; NCGC00021545-05; NCGC00261267-01; BR-35803; SMR000058311; SBI-0206904.P001; AB0068842; AM20070538; EU-0100582; FT-0626586; FT-0668920; EN300-52516; 42G963; C07018; D00332; M-2788; L000733; Q410352; SR-01000000019-2; SR-01000000019-6; SR-01000000019-11; Z1258578343; Gabapentin, European Pharmacopoeia (EP) Reference Standard; Gabapentin, United States Pharmacopeia (USP) Reference Standard; Gabapentin, Pharmaceutical Secondary Standard; Certified Reference Material
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Clinical Status |
Approved
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Disease Indication | Focal seizure | ICD-11: 8A68 | [1] | ||
PubChem CID | |||||
Formula |
C9H17NO2
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Canonical SMILES |
C1CCC(CC1)(CC(=O)O)CN
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InChI |
1S/C9H17NO2/c10-7-9(6-8(11)12)4-2-1-3-5-9/h1-7,10H2,(H,11,12)
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InChIKey |
UGJMXCAKCUNAIE-UHFFFAOYSA-N
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Click to Show/Hide the Molecular Data (Structure/Property) of This API | |||||
Structure |
<iframe style="width: 300px; height: 300px;" frameborder="0" src="https://embed.molview.org/v1/?mode=balls&cid=3446"></iframe>
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3D MOL | 2D MOL | ||||
Physicochemical Properties | Molecular Weight | 171.24 | Topological Polar Surface Area | 63.3 | |
XlogP | -1.1 | Complexity | 162 | ||
Heavy Atom Count | 12 | Rotatable Bond Count | 3 | ||
Hydrogen Bond Donor Count | 2 | Hydrogen Bond Acceptor Count | 3 | ||
Full List of Drug Formulations (DFMs) Containing This API | ||||||
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Gabapentin 100 mg capsule | Click to Show/Hide the Full List of Formulation(s): 43 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Aluminum hydroxide; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Actavis Pharma; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | McKesson; Stat Rx USA | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Aluminum hydroxide; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Bryant Ranch Prepack; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Actavis Pharma Manufacturing Pvt; Cardinal Health; DirectRX; McKesson; NCS HealthCare of KY, Inc dba Vangard Labs; NuCare Pharmaceuticals; RemedyRepack; TYA Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | American Health Packaging; Cardinal Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Actavis Pharma; Aphena Pharma Solutions-Tennessee; McKesson; PD-Rx Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Propylene glycol 1,2-distearate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Talc; Titanium dioxide; Gelatin hydrolysate (porcine skin, mw 3000); Silicon dioxide; Mannitol hexanitrate; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Gelatin | DIG Info | Mephenytoin 4-hydroxylase (EC50 = 20.5 uM) | [7] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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Sodium lauryl sulfate; Calcium carbonate; Butyl alcohol; Glyceryl behenate; Isopropyl alcohol; Ammonia; Calcium sulfate dihydrate; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Alcohol; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Calcium carbonate | DIG Info | Carbonic anhydrase IX (Ki = 8600 nM) | [9] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 15 |
DFM Info
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Sodium lauryl sulfate; Calcium carbonate; Butyl alcohol; Glyceryl dibehenate; Isopropyl alcohol; Ammonia; Calcium sulfate dihydrate; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Alcohol; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | A-S Medication Solutions; Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Calcium carbonate | DIG Info | Carbonic anhydrase IX (Ki = 8600 nM) | [9] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 16 |
DFM Info
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Butyl alcohol; Isopropyl alcohol; Magnesium stearate; Ammonia; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Croscarmellose sodium; Alcohol; Gelatin; Shellac
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Dosage Form | Oral Capsule | |||||
Company | Apotex; Carilion Materials Management; Lake Eire Medical & Surgical Supply DBA Quality Care Products; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 17 |
DFM Info
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Butyl alcohol; Isopropyl alcohol; Magnesium stearate; Ammonia; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Croscarmellose sodium; Alcohol; Gelatin, unspecified; Shellac
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health; Major Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 18 |
DFM Info
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Isopropyl alcohol; Magnesium stearate; Ammonia; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Croscarmellose sodium; Alcohol; Gelatin; Shellac
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Dosage Form | Oral Capsule | |||||
Company | Rebel Distributors | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 19 |
DFM Info
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Fd&c blue no. 2; Magnesium stearate; Mannitol; Ferric oxide yellow; Propylene glycol; Sodium hydroxide; Talc; Titanium dioxide; Gelatin, unspecified; Povidone, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 20 |
DFM Info
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Sodium lauryl sulfate; Magnesium stearate; Mannitol; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Ranbaxy Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 21 |
DFM Info
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Sodium lauryl sulfate; Butyl alcohol; Isopropyl alcohol; Ammonia; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Talc; Titanium dioxide; Alcohol; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Method Pharmaceuticals; PD-Rx Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 22 |
DFM Info
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D&c yellow no. 10; Fd&c red no. 40; Mannitol; Talc; Titanium dioxide; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 23 |
DFM Info
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D&c yellow no. 10; Fd&c red no. 40; Mannitol; Talc; Titanium dioxide; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | A-S Medication Solutions; Aphena Pharma Solutions-Tennessee; Camber Pharmaceuticals; H. J. Harkins Company; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Preferred Pharamaceuticals; Proficient Rx; RemedyRepack; TYA Pharmaceuticals; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 24 |
DFM Info
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Fd&c blue no. 1; Magnesium stearate; Propylene glycol; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Epic Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 25 |
DFM Info
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Lactose monohydrate; Fd&c blue no. 2; Propylene glycol; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Bi-Coastal Pharma International; Marksans Pharma; NuCare Pharmaceuticals; Solco Healthcare; Time Cap Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 26 |
DFM Info
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Lactose monohydrate; Fd&c blue no. 2; Propylene glycol; Talc; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Breckenridge Pharmaceutical | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 27 |
DFM Info
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Sodium lauryl sulfate; Magnesium stearate; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health; Major Pharmaceuticals; Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 28 |
DFM Info
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Lactose monohydrate; Fd&c blue no. 1; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Jiangsu Hengrui Medicine | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Drug Formulation 29 |
DFM Info
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Lactose, unspecified form; Fd&c blue no. 2; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Greenstone; Parke-Davis Div of Pfizer Inc | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Drug Formulation 30 |
DFM Info
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Sodium lauryl sulfate; Ferrosoferric oxide; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 31 |
DFM Info
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Anhydrous lactose; Sodium lauryl sulfate; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Ascend Laboratories; Avera McKennan Hospital; Cardinal Health; Clinical Solutions Wholesale; Contract Pharmacal; Department of State Health Services, Pharmacy Branch; NorthStar Rx; PD-Rx Pharmaceuticals; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 32 |
DFM Info
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Sodium lauryl sulfate; Ferrosoferric oxide; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | A-S Medication Solutions; Aphena Pharma Solutions-Tennessee; Aurobindo Pharma; Blenheim Phamacal; Lucid Pharma; NCS HealthCare of KY, Inc dba Vangard Labs; NorthStar Rx; PD-Rx Pharmaceuticals; RemedyRepack; Safecor Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 33 |
DFM Info
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Sodium lauryl sulfate; Ferrosoferric oxide; Talc; Titanium dioxide; Gelatin, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | A-S Medication Solutions; Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 34 |
DFM Info
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Mannitol; Talc; Titanium dioxide; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Aidarex Pharmaceuticals; Cipla; Clinical Solutions Wholesale; Exelan Pharmaceuticals; Lake Eire Medical & Surgical Supply DBA Quality Care Products; NuCare Pharmaceuticals; Proficient Rx; St Marys Medical Park Pharmacy; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Drug Formulation 35 |
DFM Info
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Sodium lauryl sulfate; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Akron Pharma; ScieGen Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 36 |
DFM Info
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Sodium lauryl sulfate; Talc; Titanium dioxide; Gelatin, unspecified; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 37 |
DFM Info
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Sodium lauryl sulfate; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Westminster Pharmaceuticals, LLC | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 38 |
DFM Info
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Magnesium stearate; Talc; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | PD-Rx Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 39 |
DFM Info
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Magnesium stearate; Talc; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 40 |
DFM Info
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Lactose monohydrate; Ferrosoferric oxide; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health | |||||
Drug Formulation 41 |
DFM Info
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Ferrosoferric oxide; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Dispensing Solution; Hikma Pharmaceutical; West-Ward Pharmaceticals | |||||
Drug Formulation 42 |
DFM Info
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Titanium dioxide; Gelatin
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Dosage Form | Oral Capsule | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products | |||||
Drug Formulation 43 |
DFM Info
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Talc; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | West-Ward Pharmaceticals | |||||
Gabapentin 300 mg capsule | Click to Show/Hide the Full List of Formulation(s): 54 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Aluminum hydroxide; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Actavis Pharma; NuCare Pharmaceuticals; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Aluminum hydroxide; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin, unspecified; Shellac; Starch, corn
|
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Dosage Form | Oral Capsule | |||||
Company | Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Stat Rx USA | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 7 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Actavis Pharma Manufacturing Pvt; Aphena Pharma Solutions-Tennessee; Cardinal Health; Department of State Health Services, Pharmacy Branch; NCS HealthCare of KY, Inc dba Vangard Labs; RemedyRepack; Westwood Manufacturing | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 8 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | American Health Packaging; Cardinal Health; Lake Eire Medical & Surgical Supply DBA Quality Care Products; McKesson; NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | MedVantx; NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Actavis Pharma; Aphena Pharma Solutions-Tennessee; McKesson | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Butyl alcohol; Isopropyl alcohol; Ammonia; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Talc; Titanium dioxide; Alcohol; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Method Pharmaceuticals; PD-Rx Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 15 |
DFM Info
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Fd&c yellow no. 6; Propylene glycol; Sodium hydroxide; Talc; Titanium dioxide; Fd&c red no. 3; Lecithin, soybean; Povidone; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Teva Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
FD&C red no. 3 | DIG Info | Phosphodiesterase 3A (IC50 = 0.092 uM) | [2] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [7] | |||
Soybean lecithin | DIG Info | Albendazole monooxygenase (IC50 = 6.61 mg.mL-1) | [5] | |||
Drug Formulation 16 |
DFM Info
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Sodium lauryl sulfate; Calcium carbonate; Butyl alcohol; Glyceryl behenate; Isopropyl alcohol; Ammonia; Calcium sulfate dihydrate; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Alcohol; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Calcium carbonate | DIG Info | Carbonic anhydrase IX (Ki = 8600 nM) | [9] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 17 |
DFM Info
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Sodium lauryl sulfate; Calcium carbonate; Butyl alcohol; Glyceryl dibehenate; Isopropyl alcohol; Ammonia; Calcium sulfate dihydrate; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Alcohol; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | A-S Medication Solutions; DirectRX; Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Calcium carbonate | DIG Info | Carbonic anhydrase IX (Ki = 8600 nM) | [9] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 18 |
DFM Info
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Butyl alcohol; Isopropyl alcohol; Magnesium stearate; Ammonia; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Croscarmellose sodium; Alcohol; Gelatin; Shellac
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Dosage Form | Oral Capsule | |||||
Company | Apotex; Blenheim Phamacal; Cardinal Health; Lake Eire Medical & Surgical Supply DBA Quality Care Products; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 19 |
DFM Info
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Butyl alcohol; Isopropyl alcohol; Magnesium stearate; Ammonia; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Croscarmellose sodium; Alcohol; Gelatin, unspecified; Shellac
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health; Major Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 20 |
DFM Info
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Isopropyl alcohol; Magnesium stearate; Ammonia; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Croscarmellose sodium; Alcohol; Gelatin; Shellac
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Dosage Form | Oral Capsule | |||||
Company | Rebel Distributors | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 21 |
DFM Info
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Sodium lauryl sulfate; Magnesium stearate; Mannitol; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Ranbaxy Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 22 |
DFM Info
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Fd&c blue no. 2; Magnesium stearate; Mannitol; Ferric oxide yellow; Propylene glycol; Sodium hydroxide; Talc; Titanium dioxide; Gelatin, unspecified; Povidone, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 23 |
DFM Info
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Fd&c yellow no. 6; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Fd&c red no. 3; Lecithin, soybean; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | MedVantx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
FD&C red no. 3 | DIG Info | Phosphodiesterase 3A (IC50 = 0.092 uM) | [2] | |||
Soybean lecithin | DIG Info | Albendazole monooxygenase (IC50 = 6.61 mg.mL-1) | [5] | |||
Drug Formulation 24 |
DFM Info
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Lactose monohydrate; Fd&c blue no. 1; Fd&c yellow no. 5; Fd&c yellow no. 6; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Jiangsu Hengrui Medicine | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Hydrazine yellow | DIG Info | GABA(A) receptor alpha-1 (IC50 = 13 uM) | [2] | |||
Drug Formulation 25 |
DFM Info
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Fd&c blue no. 1; Magnesium stearate; Ferric oxide yellow; Propylene glycol; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Epic Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 26 |
DFM Info
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D&c yellow no. 10; Fd&c red no. 40; Mannitol; Talc; Titanium dioxide; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 27 |
DFM Info
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D&c yellow no. 10; Fd&c red no. 40; Mannitol; Talc; Titanium dioxide; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Aphena Pharma Solutions-Tennessee; Blenheim Phamacal; Bryant Ranch Prepack; Camber Pharmaceuticals; DirectRX; Exelan Pharmaceuticals; PD-Rx Pharmaceuticals; Pharmaceutica North America; Preferred Pharamaceuticals; Proficient Rx; Raritan Pharmaceuticals; Rebel Distributors; RemedyRepack; TYA Pharmaceuticals; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 28 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Westminster Pharmaceuticals, LLC | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 29 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RedPharm | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 30 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Akron Pharma; ScieGen Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 31 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Talc; Titanium dioxide; Gelatin, unspecified; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | PD-Rx Pharmaceuticals; Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 32 |
DFM Info
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Lactose monohydrate; Fd&c blue no. 2; Ferric oxide yellow; Propylene glycol; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | AvPAK; Bi-Coastal Pharma International; MSM Repackaging ; Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 33 |
DFM Info
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Sodium lauryl sulfate; Calcium carbonate; Glyceryl behenate; Calcium sulfate dihydrate; Ferric oxide yellow; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Pharmaceutica North America | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Calcium carbonate | DIG Info | Carbonic anhydrase IX (Ki = 8600 nM) | [9] | |||
Drug Formulation 34 |
DFM Info
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Sodium lauryl sulfate; Calcium carbonate; Glyceryl dibehenate; Calcium sulfate dihydrate; Ferric oxide yellow; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | TYA Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Calcium carbonate | DIG Info | Carbonic anhydrase IX (Ki = 8600 nM) | [9] | |||
Drug Formulation 35 |
DFM Info
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Lactose monohydrate; Fd&c blue no. 2; Ferric oxide yellow; Propylene glycol; Talc; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Breckenridge Pharmaceutical | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 36 |
DFM Info
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Sodium lauryl sulfate; Magnesium stearate; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health; Major Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 37 |
DFM Info
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Sodium lauryl sulfate; Magnesium stearate; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 38 |
DFM Info
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Sodium lauryl sulfate; Magnesium stearate; Talc; Titanium dioxide; Brown iron oxide; Gelatin; Starch, pregelatinized corn
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Dosage Form | Oral Capsule | |||||
Company | Sterling Knight Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 39 |
DFM Info
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Lactose; Fd&c blue no. 2; Ferric oxide yellow; Talc; Titanium dioxide; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Drug Formulation 40 |
DFM Info
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Lactose, unspecified form; Fd&c blue no. 2; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Greenstone; Parke-Davis Div of Pfizer Inc | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Drug Formulation 41 |
DFM Info
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Lactose; Fd&c blue no. 2; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Drug Formulation 42 |
DFM Info
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Anhydrous lactose; Sodium lauryl sulfate; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 43 |
DFM Info
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Anhydrous lactose; Sodium lauryl sulfate; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RedPharm | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 44 |
DFM Info
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Anhydrous lactose; Sodium lauryl sulfate; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | A-S Medication Solutions; Aidarex Pharmaceuticals; Ascend Laboratories; Avera McKennan Hospital; Cardinal Health; Clinical Solutions Wholesale; Contract Pharmacal; Lake Eire Medical & Surgical Supply DBA Quality Care Products; NorthStar Rx; PD-Rx Pharmaceuticals; Proficient Rx; RemedyRepack; TMIG | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 45 |
DFM Info
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Anhydrous lactose; Sodium lauryl sulfate; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin, unspecified; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Preferred Pharamaceuticals; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 46 |
DFM Info
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Lactose; Sodium lauryl sulfate; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Clinical Solutions Wholesale | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 47 |
DFM Info
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Sodium lauryl sulfate; Ferric oxide yellow; Ferrosoferric oxide; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | A-S Medication Solutions; Aphena Pharma Solutions-Tennessee; Aurobindo Pharma; Lucid Pharma; MedVantx; NCS HealthCare of KY, Inc dba Vangard Labs; New Horizon Rx Group; NorthStar Rx; PD-Rx Pharmaceuticals; RemedyRepack; Safecor Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 48 |
DFM Info
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Sodium lauryl sulfate; Ferric oxide yellow; Ferrosoferric oxide; Talc; Titanium dioxide; Gelatin, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 49 |
DFM Info
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Mannitol; Talc; Titanium dioxide; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cipla; Clinical Solutions Wholesale; Lake Eire Medical & Surgical Supply DBA Quality Care Products; NuCare Pharmaceuticals; Preferred Pharamaceuticals; Proficient Rx; St Marys Medical Park Pharmacy; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Drug Formulation 50 |
DFM Info
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Mannitol; Talc; Titanium dioxide; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RedPharm | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Drug Formulation 51 |
DFM Info
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Lactose monohydrate; Ferric oxide yellow; Propylene glycol; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Marksans Pharma; NuCare Pharmaceuticals; St Marys Medical Park Pharmacy; Time Cap Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 52 |
DFM Info
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Ferric oxide yellow; Talc; Titanium dioxide; Fd&c red no. 3; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Dispensing Solution; Hikma Pharmaceutical; West-Ward Pharmaceticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C red no. 3 | DIG Info | Phosphodiesterase 3A (IC50 = 0.092 uM) | [2] | |||
Drug Formulation 53 |
DFM Info
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Magnesium stearate; Talc; Starch, corn
|
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Dosage Form | Oral Capsule | |||||
Company | Contract Pharmacal | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 54 |
DFM Info
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Talc; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | West-Ward Pharmaceticals | |||||
Gabapentin 400 mg capsule | Click to Show/Hide the Full List of Formulation(s): 40 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Aluminum hydroxide; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Actavis Pharma; St Marys Medical Park Pharmacy | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Aluminum hydroxide; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Actavis Pharma Manufacturing Pvt; Aphena Pharma Solutions-Tennessee; DirectRX; NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | American Health Packaging; Cardinal Health; Lake Eire Medical & Surgical Supply DBA Quality Care Products | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | McKesson | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 7 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 8 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Actavis Pharma; Aphena Pharma Solutions-Tennessee; Carilion Materials Management; McKesson | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 2; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health; PD-Rx Pharmaceuticals; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Fd&c blue no. 1; Mannitol; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Talc; Titanium dioxide; Silicon dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | St Marys Medical Park Pharmacy | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Butyl alcohol; Isopropyl alcohol; Ammonia; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Talc; Titanium dioxide; Alcohol; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Method Pharmaceuticals; PD-Rx Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 13 |
DFM Info
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Sodium lauryl sulfate; Calcium carbonate; Butyl alcohol; Glyceryl dibehenate; Isopropyl alcohol; Ammonia; Calcium sulfate dihydrate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Alcohol; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Calcium carbonate | DIG Info | Carbonic anhydrase IX (Ki = 8600 nM) | [9] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 14 |
DFM Info
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Sodium lauryl sulfate; Calcium carbonate; Butyl alcohol; Glyceryl dibehenate; Isopropyl alcohol; Ammonia; Calcium sulfate dihydrate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Alcohol; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Calcium carbonate | DIG Info | Carbonic anhydrase IX (Ki = 8600 nM) | [9] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 15 |
DFM Info
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Butyl alcohol; Isopropyl alcohol; Magnesium stearate; Ammonia; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Croscarmellose sodium; Alcohol; Gelatin; Shellac
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Dosage Form | Oral Capsule | |||||
Company | A-S Medication Solutions; Apotex; Blenheim Phamacal | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 16 |
DFM Info
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Butyl alcohol; Isopropyl alcohol; Magnesium stearate; Ammonia; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Croscarmellose sodium; Alcohol; Gelatin, unspecified; Shellac
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Dosage Form | Oral Capsule | |||||
Company | Bryant Ranch Prepack; Cardinal Health; Major Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 17 |
DFM Info
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Isopropyl alcohol; Magnesium stearate; Ammonia; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Titanium dioxide; Water; Croscarmellose sodium; Alcohol; Gelatin; Shellac
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Dosage Form | Oral Capsule | |||||
Company | Rebel Distributors | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [8] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 18 |
DFM Info
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Sodium lauryl sulfate; Magnesium stearate; Mannitol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Ranbaxy Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 19 |
DFM Info
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Fd&c blue no. 2; Magnesium stearate; Mannitol; Ferric oxide yellow; Propylene glycol; Sodium hydroxide; Talc; Titanium dioxide; Gelatin, unspecified; Povidone, unspecified; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 20 |
DFM Info
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Sodium lauryl sulfate; Fd&c blue no. 1; Fd&c yellow no. 6; Magnesium stearate; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cardinal Health; Major Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 21 |
DFM Info
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Sodium lauryl sulfate; Fd&c blue no. 1; Fd&c yellow no. 6; Magnesium stearate; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Physicians Total Care; Stat Rx USA | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 22 |
DFM Info
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Fd&c blue no. 1; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Propylene glycol; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Epic Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 23 |
DFM Info
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Lactose monohydrate; Fd&c blue no. 1; Fd&c yellow no. 5; Fd&c yellow no. 6; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Jiangsu Hengrui Medicine | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Hydrazine yellow | DIG Info | GABA(A) receptor alpha-1 (IC50 = 13 uM) | [2] | |||
Drug Formulation 24 |
DFM Info
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D&c yellow no. 10; Fd&c red no. 40; Mannitol; Talc; Titanium dioxide; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Aphena Pharma Solutions-Tennessee; Blenheim Phamacal; Bryant Ranch Prepack; Camber Pharmaceuticals; Exelan Pharmaceuticals; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Medsource Pharmaceuticals; Preferred Pharamaceuticals; Proficient Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 25 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Akron Pharma; ScieGen Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 26 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Talc; Titanium dioxide; Gelatin, unspecified; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 27 |
DFM Info
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Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Westminster Pharmaceuticals, LLC | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 28 |
DFM Info
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Sodium lauryl sulfate; Calcium carbonate; Glyceryl behenate; Calcium sulfate dihydrate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Calcium carbonate | DIG Info | Carbonic anhydrase IX (Ki = 8600 nM) | [9] | |||
Drug Formulation 29 |
DFM Info
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Lactose monohydrate; Fd&c blue no. 2; Ferric oxide yellow; Propylene glycol; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | AvPAK; Bi-Coastal Pharma International; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Marksans Pharma; Solco Healthcare; Time Cap Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 30 |
DFM Info
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Lactose monohydrate; Fd&c blue no. 2; Ferric oxide red; Ferric oxide yellow; Propylene glycol; Talc; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Breckenridge Pharmaceutical | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [5] | |||
Drug Formulation 31 |
DFM Info
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Fd&c blue no. 2; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Fd&c red no. 3; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Hikma Pharmaceutical | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
FD&C red no. 3 | DIG Info | Phosphodiesterase 3A (IC50 = 0.092 uM) | [2] | |||
Drug Formulation 32 |
DFM Info
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Fd&c blue no. 2; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Fd&c red no. 3; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | West-Ward Pharmaceticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
FD&C red no. 3 | DIG Info | Phosphodiesterase 3A (IC50 = 0.092 uM) | [2] | |||
Drug Formulation 33 |
DFM Info
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D&c yellow no. 10; Fd&c red no. 40; Talc; Titanium dioxide; Mannitol hexanitrate; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 34 |
DFM Info
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Lactose, unspecified form; Fd&c blue no. 2; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Greenstone; Parke-Davis Div of Pfizer Inc | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Drug Formulation 35 |
DFM Info
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Lactose; Fd&c blue no. 2; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Stat Rx USA | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Drug Formulation 36 |
DFM Info
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Anhydrous lactose; Sodium lauryl sulfate; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | A-S Medication Solutions; Aidarex Pharmaceuticals; Ascend Laboratories; Avera McKennan Hospital; Cardinal Health; Contract Pharmacal; NorthStar Rx; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 37 |
DFM Info
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Anhydrous lactose; Sodium lauryl sulfate; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Gelatin, unspecified; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Preferred Pharamaceuticals; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 38 |
DFM Info
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Sodium lauryl sulfate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Talc; Titanium dioxide; Gelatin; Shellac; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Aphena Pharma Solutions-Tennessee; Aurobindo Pharma; Lucid Pharma; NCS HealthCare of KY, Inc dba Vangard Labs; NorthStar Rx; RemedyRepack; Safecor Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 39 |
DFM Info
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Mannitol; Talc; Titanium dioxide; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | Cipla; Lake Eire Medical & Surgical Supply DBA Quality Care Products; NuCare Pharmaceuticals; Preferred Pharamaceuticals; Proficient Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Drug Formulation 40 |
DFM Info
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Talc; Starch, corn
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Dosage Form | Oral Capsule | |||||
Company | West-Ward Pharmaceticals | |||||
Gabapentin 600 mg tablet | Click to Show/Hide the Full List of Formulation(s): 59 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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Glyceryl behenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Hypromellose; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose; Hydroxypropyl cellulose, low substituted; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Rebel Distributors | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Hypromellose | DIG Info | Cytochrome P450 3A5 (IC50 = 19.4 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 2 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Poloxamer 407; Silicon dioxide; Copovidone; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Method Pharmaceuticals; PD-Rx Pharmaceuticals; Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Poloxamer 407; Silicon dioxide; Copovidone k25-31; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycol, unspecified
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Dosage Form | Oral Tablet | |||||
Company | Akron Pharma; ScieGen Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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Glyceryl dibehenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose (type h); Hydroxypropyl cellulose, low substituted; Hypromelloses; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 5 |
DFM Info
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Glyceryl dibehenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose; Hydroxypropyl cellulose, low substituted; Hypromelloses; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 6 |
DFM Info
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Glyceryl dibehenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Low-substituted hydroxypropyl cellulose, unspecified; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 7 |
DFM Info
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Glyceryl dibehenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose (type h); Hydroxypropyl cellulose, low substituted; Hypromellose 2208 (100 mpa.s); Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Clinical Solutions Wholesale | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 8 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose (120000 mw); Hypromellose 2910 (3 mpa.s); Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Liberty Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose (type h); Hypromellose 2910 (3 mpa.s); Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | AvPAK | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | A-S Medication Solutions; Camber Pharmaceuticals; Cipla; Contract Pharmacal; Lake Eire Medical & Surgical Supply DBA Quality Care Products; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose; Hypromellose 2910 (3 mpa.s); Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Aphena Pharma Solutions-Tennessee | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Poloxamer 407; Polyvinyl alcohol; Copovidone k25-31; Hydroxypropyl cellulose (type h); Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | ACI Healthcare USA; Lake Eire Medical & Surgical Supply DBA Quality Care Products; NuCare Pharmaceuticals; Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Poloxamer 407; Polyvinyl alcohol; Copovidone; Hydroxypropyl cellulose; Hydroxypropyl cellulose, low substituted; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Allied Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 15 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | DirectRX; RxChange | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 16 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Poloxamer 407; Silicon dioxide; Copovidone k25-31; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Polyethylene glycol, unspecified
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Dosage Form | Oral Tablet | |||||
Company | Westminster Pharmaceuticals, LLC | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 17 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Poloxamer 407; Silicon dioxide; Copovidone k25-31; Crospovidone, unspecified; Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Polyethylene glycol, unspecified
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Dosage Form | Oral Tablet | |||||
Company | PD-Rx Pharmaceuticals; Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 18 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Poloxamer 407; Povidone; Copovidone; Hydroxypropyl cellulose, low substituted
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Dosage Form | Oral Tablet | |||||
Company | Cadila Healthcare; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 19 |
DFM Info
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Sodium lauryl sulfate; Glyceryl dibehenate; Magnesium stearate; Calcium phosphate, dibasic, dihydrate; Talc; Silicon dioxide
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Dosage Form | 24 HR Extended Release Tablet | |||||
Company | GlaxoSmithKline | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 20 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polysorbate 80; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Preferred Pharamaceuticals; Proficient Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 21 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polysorbate 80; Crospovidone, unspecified; Hydroxypropyl cellulose, unspecified; Hypromellose, unspecified; Polyethylene glycol, unspecified
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Dosage Form | Oral Tablet | |||||
Company | Exelan Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 22 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Poloxamer 407; Copovidone; Hydroxypropyl cellulose (1200000 mw); Polyethylene glycol, unspecified; Polyvinyl alcohol, unspecified
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Dosage Form | Oral Tablet | |||||
Company | Preferred Pharamaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 23 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polysorbate 80; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Polyethylene glycol, unspecified
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Dosage Form | Oral Tablet | |||||
Company | Preferred Pharamaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 24 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polysorbate 80; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 25 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Poloxamer 407; Copovidone; Low-substituted hydroxypropyl cellulose, unspecified; Povidone, unspecified
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging; Cardinal Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 26 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Poloxamer 407; Copovidone k25-31; Hydroxypropyl cellulose, low substituted; Povidones
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Dosage Form | Oral Tablet | |||||
Company | BluePoint Laboratories; McKesson | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 27 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Poloxamer 407; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose, unspecified
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Dosage Form | Oral Tablet | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 28 |
DFM Info
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Calcium stearate; Fd&c blue no. 2; Ferric oxide yellow; Titanium dioxide; Crospovidone; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 29 |
DFM Info
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Calcium stearate; Fd&c blue no. 2; Ferric oxide yellow; Titanium dioxide; Crospovidone; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging; Cardinal Health; McKesson; Proficient Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 30 |
DFM Info
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Calcium stearate; Fd&c blue no. 2; Ferric oxide yellow; Titanium dioxide; Crospovidone; Hydroxypropyl cellulose (type h); Polyethylene glycol 8000
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Dosage Form | Oral Tablet | |||||
Company | Actavis Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 31 |
DFM Info
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Calcium stearate; Fd&c blue no. 2; Ferric oxide yellow; Titanium dioxide; Crospovidone; Hydroxypropyl cellulose; Hypromelloses; Polyethylene glycol
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Dosage Form | Oral Tablet | |||||
Company | Cardinal Health; McKesson; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 32 |
DFM Info
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Calcium stearate; Fd&c blue no. 2; Ferric oxide yellow; Titanium dioxide; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 2 | DIG Info | Adenosine receptor A3 (IC50 = 1 uM) | [2] | |||
Drug Formulation 33 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Hypromellose; Poloxamer 407; Polysorbate 80; Copovidone; Polyethylene glycol; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Contract Pharmacal; Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Hypromellose | DIG Info | Cytochrome P450 3A5 (IC50 = 19.4 uM) | [7] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 34 |
DFM Info
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Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Polyethylene glycol 3350; Polyvinyl alcohol; Copovidone k25-31; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 35 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone; Hypromellose, unspecified; Polyethylene glycol, unspecified; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Glenmark Pharmaceutials; Preferred Pharamaceuticals; St Marys Medical Park Pharmacy | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 36 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone k25-31; Hypromelloses; Polyethylene glycol; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | H. J. Harkins Company | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 37 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone k25-31; Hypromellose, unspecified; Polyethylene glycol, unspecified; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Bryant Ranch Prepack; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 38 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone k25-31; Hypromelloses; Polyethylene glycols; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | A-S Medication Solutions; Blenheim Phamacal; Medsource Pharmaceuticals; NuCare Pharmaceuticals; PD-Rx Pharmaceuticals; Proficient Rx; Rebel Distributors; RemedyRepack; TYA Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 39 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone k25-31; Hypromelloses; Polyethylene glycols; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 40 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone; Hypromelloses; Polyethylene glycol; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 41 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone; Hypromelloses; Polyethylene glycols; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Aidarex Pharmaceuticals; NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 42 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone; Hypromelloses; Polyethylene glycol; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 43 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Polyethylene glycol 3350; Copovidone; Hypromellose, unspecified; Polyethylene glycol, unspecified; Polyvinyl alcohol, unspecified
|
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Dosage Form | Oral Tablet | |||||
Company | Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 44 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Polyethylene glycol 3350; Copovidone k25-31; Hypromellose, unspecified; Polyethylene glycol, unspecified; Polyvinyl alcohol, unspecified
|
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Dosage Form | Oral Tablet | |||||
Company | Depomed | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 45 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Water; Poloxamer 407; Candelilla wax; Copovidone k25-31; Hydroxypropyl cellulose (type h); Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Parke-Davis Div of Pfizer Inc | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 46 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Water; Poloxamer 407; Candelilla wax; Hydroxypropyl cellulose (type h); Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Greenstone | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 47 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Crospovidone; Cellulose, microcrystalline; Copovidone; Hydroxypropyl cellulose (type h); Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | NorthStar Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 48 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Crospovidone; Copovidone; Hydroxypropyl cellulose (type h); Microcrystalline cellulose; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Aurobindo Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 49 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Crospovidone; Cellulose, microcrystalline; Copovidone; Hydroxypropyl cellulose; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 50 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Crospovidone; Cellulose, microcrystalline; Copovidone k25-31; Hydroxypropyl cellulose (type h); Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Aidarex Pharmaceuticals; Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 51 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Poloxamer 407; Copovidone; Hydroxypropyl cellulose (type h); Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Ascend Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 52 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Titanium dioxide; Copovidone; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycol 8000
|
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Dosage Form | Oral Tablet | |||||
Company | Apotex; NuCare Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 53 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Cellulose, microcrystalline; Copovidone k25-31; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (type h); Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 54 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Titanium dioxide; Copovidone; Hydroxypropyl cellulose; Hypromelloses; Polyethylene glycol 8000
|
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Dosage Form | Oral Tablet | |||||
Company | Apotex | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 55 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Copovidone; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (1200000 mw); Microcrystalline cellulose; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Preferred Pharamaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 56 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Titanium dioxide; Copovidone k25-31; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycol 8000
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Dosage Form | Oral Tablet | |||||
Company | Golden State Medical Supply | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 57 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Cellulose, microcrystalline; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products | |||||
Drug Formulation 58 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Microcrystalline cellulose; Polyethylene glycol 8000
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Dosage Form | Oral Tablet | |||||
Company | Teva Pharmaceuticals | |||||
Drug Formulation 59 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Cellulose, microcrystalline; Polyethylene glycol
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack; Stat Rx USA | |||||
Gabapentin 800 mg tablet | Click to Show/Hide the Full List of Formulation(s): 53 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Glyceryl behenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Hypromellose; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose; Hydroxypropyl cellulose, low substituted; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Rebel Distributors; Stat Rx USA | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Hypromellose | DIG Info | Cytochrome P450 3A5 (IC50 = 19.4 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Poloxamer 407; Silicon dioxide; Copovidone; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | Method Pharmaceuticals; PD-Rx Pharmaceuticals; Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Poloxamer 407; Silicon dioxide; Copovidone k25-31; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycol, unspecified
|
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Dosage Form | Oral Tablet | |||||
Company | Akron Pharma; ScieGen Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Glyceryl dibehenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose (type h); Hydroxypropyl cellulose, low substituted; Hypromelloses; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Clinical Solutions Wholesale; Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Glyceryl dibehenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose; Hydroxypropyl cellulose, low substituted; Hypromelloses; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Glyceryl dibehenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Low-substituted hydroxypropyl cellulose, unspecified; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Glyceryl behenate; Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polyethylene glycol 400; Polysorbate 80; Hydroxypropyl cellulose; Hydroxypropyl cellulose, low substituted; Hypromelloses; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose; Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose (120000 mw); Hypromellose 2910 (3 mpa.s); Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | Liberty Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose (type h); Hypromellose 2910 (3 mpa.s); Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | AvPAK | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | A-S Medication Solutions; Aidarex Pharmaceuticals; Camber Pharmaceuticals; Cipla; Contract Pharmacal; Proficient Rx; St Marys Medical Park Pharmacy | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose; Hypromellose 2910 (3 mpa.s); Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | Aphena Pharma Solutions-Tennessee | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Poloxamer 407; Silicon dioxide; Copovidone; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Polyethylene glycol, unspecified
|
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Dosage Form | Oral Tablet | |||||
Company | Atlantic Biologicals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Poloxamer 407; Silicon dioxide; Copovidone k25-31; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Polyethylene glycol, unspecified
|
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Dosage Form | Oral Tablet | |||||
Company | Westminster Pharmaceuticals, LLC | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 15 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Poloxamer 407; Polyvinyl alcohol; Copovidone; Hydroxypropyl cellulose; Hydroxypropyl cellulose, low substituted; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | Allied Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 16 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose (type h); Hypromelloses
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 17 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Poloxamer 407; Silicon dioxide; Copovidone k25-31; Crospovidone, unspecified; Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Polyethylene glycol, unspecified
|
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Dosage Form | Oral Tablet | |||||
Company | Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 18 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Titanium dioxide; Crospovidone; Polysorbate 80; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 19 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Poloxamer 407; Povidone; Copovidone; Hydroxypropyl cellulose, low substituted
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Dosage Form | Oral Tablet | |||||
Company | Cadila Healthcare; DirectRX; PD-Rx Pharmaceuticals; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 20 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Poloxamer 407; Polyvinyl alcohol; Copovidone k25-31; Hydroxypropyl cellulose (type h); Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | ACI Healthcare USA; Lake Eire Medical & Surgical Supply DBA Quality Care Products; RemedyRepack; Solco Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 21 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Mannitol; Talc; Crospovidone; Poloxamer 407; Hydroxypropyl cellulose
|
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Dosage Form | Oral Tablet | |||||
Company | UDL Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 22 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polysorbate 80; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Preferred Pharamaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 23 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Titanium dioxide; Polysorbate 80; Crospovidone, unspecified; Hydroxypropyl cellulose, unspecified; Hypromellose, unspecified; Polyethylene glycol, unspecified
|
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Dosage Form | Oral Tablet | |||||
Company | Exelan Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 24 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Poloxamer 407; Copovidone; Low-substituted hydroxypropyl cellulose, unspecified; Povidone, unspecified
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging; Cardinal Health | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 25 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Poloxamer 407; Copovidone k25-31; Hydroxypropyl cellulose, low substituted; Povidones
|
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Dosage Form | Oral Tablet | |||||
Company | BluePoint Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 26 |
DFM Info
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Magnesium stearate; Mannitol; Talc; Poloxamer 407; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose, unspecified
|
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Dosage Form | Oral Tablet | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 27 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Hypromellose; Poloxamer 407; Polysorbate 80; Copovidone; Polyethylene glycol; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Hypromellose | DIG Info | Cytochrome P450 3A5 (IC50 = 19.4 uM) | [7] | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 28 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone; Hypromellose, unspecified; Polyethylene glycol, unspecified; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Contract Pharmacal; Glenmark Pharmaceutials; NuCare Pharmaceuticals; Preferred Pharamaceuticals; RemedyRepack; St Marys Medical Park Pharmacy | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 29 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone k25-31; Hypromelloses; Polyethylene glycol; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | H. J. Harkins Company | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 30 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone k25-31; Hypromellose, unspecified; Polyethylene glycol, unspecified; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Bryant Ranch Prepack; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 31 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone k25-31; Hypromelloses; Polyethylene glycols; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Blenheim Phamacal; Proficient Rx; Rebel Distributors; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 32 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone k25-31; Hypromelloses; Polyethylene glycols; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 33 |
DFM Info
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Magnesium stearate; Talc; Titanium dioxide; Water; Poloxamer 407; Polysorbate 80; Copovidone; Hypromelloses; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 34 |
DFM Info
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Magnesium stearate; Talc; Crospovidone; Poloxamer 407; Copovidone; Corn starch 3-e-dodecenyl succinic anhydride modified; Hydroxypropyl cellulose
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Dosage Form | Oral Tablet | |||||
Company | Hikma Pharmaceutical | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 35 |
DFM Info
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Calcium stearate; Ferrosoferric oxide; Titanium dioxide; Crospovidone; Polyethylene glycol 400; Hydroxypropyl cellulose (type h); Hypromellose, unspecified; Polyethylene glycol 8000
|
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Dosage Form | Oral Tablet | |||||
Company | Actavis Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [5] | |||
Drug Formulation 36 |
DFM Info
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Magnesium stearate; Talc; Water; Poloxamer 407; Candelilla wax; Copovidone k25-31; Hydroxypropyl cellulose (type h); Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Parke-Davis Div of Pfizer Inc | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 37 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Water; Poloxamer 407; Candelilla wax; Hydroxypropyl cellulose (type h); Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Greenstone | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 38 |
DFM Info
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Magnesium stearate; Talc; Crospovidone; Cellulose, microcrystalline; Copovidone; Hydroxypropyl cellulose (type h); Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | NorthStar Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 39 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Crospovidone; Copovidone; Hydroxypropyl cellulose (type h); Microcrystalline cellulose; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Aurobindo Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 40 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Crospovidone; Cellulose, microcrystalline; Copovidone; Hydroxypropyl cellulose; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 41 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Crospovidone; Cellulose, microcrystalline; Copovidone k25-31; Hydroxypropyl cellulose (type h); Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Aidarex Pharmaceuticals; Bryant Ranch Prepack; Proficient Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 42 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Poloxamer 407; Copovidone; Hydroxypropyl cellulose (type h); Starch, corn
|
|||||
Dosage Form | Oral Tablet | |||||
Company | Ascend Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Poloxamer 407 | DIG Info | Albendazole monooxygenase (EC50 = 32.8 uM) | [7] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 43 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Crospovidone; Cellulose, microcrystalline; Copovidone; Hydroxypropyl cellulose; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 44 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Calcium stearate; Ferrosoferric oxide; Titanium dioxide; Crospovidone; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 45 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Calcium stearate; Ferrosoferric oxide; Titanium dioxide; Crospovidone; Hydroxypropyl cellulose; Hypromelloses; Polyethylene glycol
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 46 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Calcium stearate; Ferric oxide yellow; Titanium dioxide; Crospovidone; Hydroxypropyl cellulose; Hypromelloses; Polyethylene glycol
|
|||||
Dosage Form | Oral Tablet | |||||
Company | McKesson | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 47 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Titanium dioxide; Copovidone; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycol 8000
|
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Dosage Form | Oral Tablet | |||||
Company | Apotex | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 48 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Cellulose, microcrystalline; Copovidone k25-31; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (type h); Starch, corn
|
|||||
Dosage Form | Oral Tablet | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 49 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Calcium stearate; Ferrosoferric oxide; Titanium dioxide; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
Drug Formulation 50 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Calcium stearate; Ferrosoferric oxide; Titanium dioxide; Crospovidone (15 mpa.s at 5%); Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | PD-Rx Pharmaceuticals | |||||
Drug Formulation 51 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Cellulose, microcrystalline; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products | |||||
Drug Formulation 52 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Microcrystalline cellulose; Polyethylene glycol 8000
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Dosage Form | Oral Tablet | |||||
Company | Teva Pharmaceuticals; Unit Dose Services | |||||
Drug Formulation 53 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Cellulose, microcrystalline; Polyethylene glycol 8000
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Dosage Form | Oral Tablet | |||||
Company | Clinical Solutions Wholesale | |||||
Gabapentin 300 mg tablet | Click to Show/Hide the Full List of Formulation(s): 3 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Glyceryl dibehenate; Magnesium stearate; Dibasic calcium phosphate dihydrate; Talc; Silicon dioxide
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Dosage Form | Extended Release Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Talc; Titanium dioxide; Lecithin, soybean; Polyethylene glycol 3350; Copovidone k25-31; Hypromellose, unspecified; Microcrystalline cellulose; Polyethylene glycol, unspecified; Polyvinyl alcohol, unspecified
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Dosage Form | Oral Tablet | |||||
Company | Depomed | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Soybean lecithin | DIG Info | Albendazole monooxygenase (IC50 = 6.61 mg.mL-1) | [5] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Titanium dioxide; Copovidone k25-31; Hydroxypropyl cellulose (type h); Hypromellose 2910 (15 mpa.s); Polyethylene glycol 8000
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Dosage Form | Oral Tablet | |||||
Company | Apotex | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Gabapentin Enacarbil 300mg extended release tablet | Click to Show/Hide the Full List of Formulation(s): 1 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Colloidal Silicon Dioxide; Dibasic Calcium Phosphate Dihydrate; Glyceryl Behenate; Magnesium Stearate; Sodium Lauryl Sulfate; Talc
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Dosage Form | Extended Release Tablet | |||||
Company | Arbor Pharms | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Gabapentin Enacarbil 600mg extended release tablet | Click to Show/Hide the Full List of Formulation(s): 1 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Colloidal Silicon Dioxide; Dibasic Calcium Phosphate Dihydrate; Glyceryl Behenate; Magnesium Stearate; Sodium Lauryl Sulfate; Talc
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Dosage Form | Extended Release Tablet | |||||
Company | Arbor Pharms | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Gabapentin 100 mg tablet | Click to Show/Hide the Full List of Formulation(s): 1 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Titanium dioxide; Copovidone k25-31; Hydroxypropyl cellulose (type h); Hypromellose 2910 (15 mpa.s); Polyethylene glycol 8000
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Dosage Form | Oral Tablet | |||||
Company | Apotex | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Gabapentin 400 mg tablet | Click to Show/Hide the Full List of Formulation(s): 1 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Magnesium stearate; Titanium dioxide; Copovidone k25-31; Hydroxypropyl cellulose (type h); Hypromellose 2910 (15 mpa.s); Polyethylene glycol 8000
|
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Dosage Form | Oral Tablet | |||||
Company | Apotex | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
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