Details of the Active Pharmaceutical Ingredient (API)

General Information of API (ID: D00445)
Name	Montelukast
Synonyms	Click to Show/Hide the Synonyms of This API montelukast; 158966-92-8; Singulair; UNII-MHM278SD3E; (R-(E))-1-(((1-(3-(2-(7-Chloro-2-quinolinyl)ethenyl)phenyl)-3-(2-(1-hydroxy-1-methylethyl)phenyl)propyl)thio)methyl)cyclopropaneacetic acid; CHEMBL787; MHM278SD3E; CHEBI:50730; Cyclopropaneacetic acid, 1-((((1R)-1-(3-((1E)-2-(7-chloro-2-quinolinyl)ethenyl)phenyl)-3-(2-(1-hydroxy-1-methylethyl)phenyl)propyl)thio)methyl)-; Montelukast [INN:BAN]; 142522-28-9; Aerokast; Brondilat (TN); 1-[[[(1 R)-1-[3-[(1E)-2-(7-chloro-2-quinolinyl)ethenyl] phenyl]-3-[2-(1-hydroxy-1-methylethyl)phenyl]propyl]sulfanyl]methyl]cyclopropaneacetic acid; 2-[1-({[(1R)-1-{3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl}-3-[2-(2-hydroxypropan-2-yl)phenyl]propyl]sulfanyl}methyl)cyclopropyl]acetic acid; Montelukast (INN); SR-01000763441; HSDB 7582; 1-((((1R)-1-(3-((1E)-2-(7-Chloro-2-quinolinyl)ethenyl)phenyl)-3-(2-(1-hydroxy-1-methylethyl)phenyl)propyl)thio)methyl)cyclopropaneacetic acid; SCHEMBL4486; SCHEMBL4487; {1-[({(1R)-1-{3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl}-3-[2-(1-hydroxy-1-methylethyl)phenyl]propyl}sulfanyl)methyl]cyclopropyl}acetic acid; BIDD:GT0394; GTPL3340; DTXSID9023334; CHEBI:94710; HMS2089D07; HMS3715N13; HMS3886L03; ACT04773; ZINC3831151; BDBM50052024; HY-13315A; AKOS025310659; CCG-221186; DB00471; SB19081; NCGC00188977-01; {1-[({(1R)-1-{3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl}-3-[2-(2-hydroxypropan-2-yl)phenyl]propyl}sulfanyl)methyl]cyclopropyl}acetic acid; 2-[1-[[(1R)-1-[3-[(E)-2-(7-chloro-2-quinolyl)vinyl]phenyl]-3-[2-(1-hydroxy-1-methyl-ethyl)phenyl]propyl]sulfanylmethyl]cyclopropyl]acetic acid; Cyclopropaneacetic acid, 1-(((1-(3-(2-(7-chloro-2-quinolinyl)ethenyl)phenyl)-3-(2-(1-hydroxy-1-methylethyl)phenyl)propyl)thio)methyl)-, (R-(E))-; CS-0002595; 5306-EP2270008A1; 5306-EP2276739A1; 5306-EP2280006A1; 5306-EP2281813A1; 5306-EP2281815A1; 5306-EP2281819A1; 5306-EP2284166A1; 5306-EP2287154A1; 5306-EP2288595A2; 5306-EP2292617A1; 5306-EP2292619A1; 5306-EP2295409A1; 5306-EP2298415A1; 5306-EP2301933A1; 5306-EP2305640A2; 5306-EP2305659A1; 5306-EP2308562A2; 5306-EP2311818A1; 5306-EP2311827A1; 5306-EP2314590A1; C07482; D08229; AB01275454-01; 522M289; Q417767; SR-01000763441-3; SR-01000763441-5; BRD-K99673372-001-01-9; 1-[[[(R)-3-[2-(1-Hydroxy-1-methylethyl)phenyl]-1-[3-[2-(7-chloroquinoline-2-yl)ethenyl]phenyl]propyl]thio]methyl]cyclopropane-1-acetic acid; 1124196-02-6; r-(e)-1-[[[1-[3-[2-(7-chloro-2-quinolinyl)ethenyl]phenyl]-3-[2-(1-hydroxy-1-methylethyl)phenyl]propyl]thio]methyl]cyclopropaneacetic acid
Clinical Status	Approved
Disease Indication	Asthma		ICD-11: CA23	[1]
PubChem CID	5281040
Formula	C35H36ClNO3S
Canonical SMILES	CC(C)(C1=CC=CC=C1CC[C@H](C2=CC=CC(=C2)/C=C/C3=NC4=C(C=CC(=C4)Cl)C=C3)SCC5(CC5)CC(=O)O)O
InChI	1S/C35H36ClNO3S/c1-34(2,40)30-9-4-3-7-25(30)13-17-32(41-23-35(18-19-35)22-33(38)39)27-8-5-6-24(20-27)10-15-29-16-12-26-11-14-28(36)21-31(26)37-29/h3-12,14-16,20-21,32,40H,13,17-19,22-23H2,1-2H3,(H,38,39)/b15-10+/t32-/m1/s1
InChIKey	UCHDWCPVSPXUMX-TZIWLTJVSA-N
	Click to Show/Hide the Molecular Data (Structure/Property) of This API
Structure	<iframe style="width: 300px; height: 300px;" frameborder="0" src="https://embed.molview.org/v1/?mode=balls&cid=5281040"></iframe>
Structure	3D MOL		2D MOL
Physicochemical Properties	Molecular Weight	586.2	Topological Polar Surface Area	95.7
	XlogP	7.7	Complexity	891
	Heavy Atom Count	41	Rotatable Bond Count	12
	Hydrogen Bond Donor Count	2	Hydrogen Bond Acceptor Count	5

Full List of Drug Formulations (DFMs) Containing This API
Montelukast 4 mg tablet			Click to Show/Hide the Full List of Formulation(s): 24 Formulation(s)
Drug Formulation 1	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Fd&c red no. 40; Maltodextrin; Aspartame; Benzyl alcohol; Magnesium stearate; Mannitol; Lactic acid, unspecified form; Ferric oxide red; Sucrose; Croscarmellose sodium; Lecithin, soybean; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Sandoz
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Allura red AC dye	DIG Info	Solute carrier SLCO2B1 (Ki = 4.7 uM)	[2]
	Benzyl alcohol	DIG Info	Indoleamine 2,3-dioxygenase 1 (IC50 = 1400 nM)	[3]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Allura red AC dye	DIG Info	Solute carrier SLCO2B1 (Ki = 2.59 uM)	[5]
	Lactic acid	DIG Info	Fetal lung MRC5 cells (IC50 = 23930 nM)	[6]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Dextrin	DIG Info	Colon cancer Caco-2 cells (Inhibition ratio > 55 %)	[8]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Soybean lecithin	DIG Info	Albendazole monooxygenase (IC50 = 6.61 mg.mL-1)	[9]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 2	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium lauryl sulfate; Fd&c red no. 40; Aspartame; Magnesium stearate; Mannitol; Croscarmellose sodium; Silicon dioxide; Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	Mylan Pharamceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Allura red AC dye	DIG Info	Solute carrier SLCO2B1 (Ki = 4.7 uM)	[2]
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Allura red AC dye	DIG Info	Solute carrier SLCO2B1 (Ki = 2.59 uM)	[5]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 3	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Sucralose; Mannitol; Butylated hydroxyanisole; Ferric oxide red; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Chewable Tablet
Company	Kremers Urban Pharmaceuticals Inc.
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sucralose	DIG Info	Carbonic anhydrase II (Ki = 300 nM)	[10]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Butylhydroxyanisole	DIG Info	Prostaglandin G/H synthase 2 (IC50 = 2.6 uM)	[2]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 4	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Sucralose; Mannitol; Butylated hydroxyanisole; Ferric oxide red; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Chewable Tablet
Company	AvKARE
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sucralose	DIG Info	Carbonic anhydrase II (Ki = 300 nM)	[10]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Butylhydroxyanisole	DIG Info	Prostaglandin G/H synthase 2 (IC50 = 2.6 uM)	[2]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 5	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Sucralose; Mannitol; Butylated hydroxyanisole; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	AvPAK
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sucralose	DIG Info	Carbonic anhydrase II (Ki = 300 nM)	[10]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Butylhydroxyanisole	DIG Info	Prostaglandin G/H synthase 2 (IC50 = 2.6 uM)	[2]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 6	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium lauryl sulfate; Maltodextrin; Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Hydroxypropyl cellulose (type h); Sodium starch glycolate type a potato; Starch, corn
Dosage Form	Chewable Tablet
Company	Carilion Materials Management; Teva Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Dextrin	DIG Info	Colon cancer Caco-2 cells (Inhibition ratio > 55 %)	[8]
Drug Formulation 7	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium lauryl sulfate; Maltodextrin; Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Hydroxypropyl cellulose; Sodium starch glycolate type a potato; Starch, corn
Dosage Form	Chewable Tablet
Company	Physicians Total Care
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Dextrin	DIG Info	Colon cancer Caco-2 cells (Inhibition ratio > 55 %)	[8]
Drug Formulation 8	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium lauryl sulfate; Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Colloidal silicon dioxide; Hydroxypropyl cellulose (type el)
Dosage Form	Chewable Tablet
Company	Hangzhou Minsheng Binjiang Pharm
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 9	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Strawberry
Dosage Form	Chewable Tablet
Company	Jubilant Cadista Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 10	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Edetate disodium; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Macleods Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 11	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry
Dosage Form	Chewable Tablet
Company	A-S Medication Solutions; NuCare Pharmaceuticals; PD-Rx Pharmaceuticals; Proficient Rx; Torrent Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 12	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Dr Reddy's Laboratories
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 13	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Camber Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 14	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	A-S Medication Solutions; Par Pharmaceutical
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 15	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Citron Pharma; Lucid Pharma
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 16	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cherry; Hydroxypropyl cellulose (type h); Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	Aurobindo Pharma
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 17	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose
Dosage Form	Chewable Tablet
Company	Greenstone
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 18	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline
Dosage Form	Chewable Tablet
Company	American Health Packaging; Apotex; Bryant Ranch Prepack
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 19	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Ajanta Pharmaceutical; Proficient Rx
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 20	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	ASE Direct; Bionpharma; Recipharm Pharmaservices; WellSpring Pharmaceutical
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 21	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose
Dosage Form	Chewable Tablet
Company	A-S Medication Solutions; Bryant Ranch Prepack
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 22	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Hydroxypropyl cellulose (1200000 mw); Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	Preferred Pharamaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 23	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cherry; Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	Preferred Pharamaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 24	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sucralose; Magnesium stearate; Mannitol; Ferric oxide red; Cellulose, microcrystalline; Copovidone k25-31; Sodium starch glycolate type a potato
Dosage Form	Chewable Tablet
Company	West-Ward Pharmaceticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sucralose	DIG Info	Carbonic anhydrase II (Ki = 300 nM)	[10]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Montelukast 5 mg tablet			Click to Show/Hide the Full List of Formulation(s): 27 Formulation(s)
Drug Formulation 1	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Fd&c red no. 40; Maltodextrin; Aspartame; Benzyl alcohol; Magnesium stearate; Mannitol; Lactic acid, unspecified form; Ferric oxide red; Sucrose; Croscarmellose sodium; Lecithin, soybean; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Sandoz
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Allura red AC dye	DIG Info	Solute carrier SLCO2B1 (Ki = 4.7 uM)	[2]
	Benzyl alcohol	DIG Info	Indoleamine 2,3-dioxygenase 1 (IC50 = 1400 nM)	[3]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Allura red AC dye	DIG Info	Solute carrier SLCO2B1 (Ki = 2.59 uM)	[5]
	Lactic acid	DIG Info	Fetal lung MRC5 cells (IC50 = 23930 nM)	[6]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Dextrin	DIG Info	Colon cancer Caco-2 cells (Inhibition ratio > 55 %)	[8]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Soybean lecithin	DIG Info	Albendazole monooxygenase (IC50 = 6.61 mg.mL-1)	[9]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 2	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium lauryl sulfate; Fd&c red no. 40; Aspartame; Magnesium stearate; Mannitol; Croscarmellose sodium; Silicon dioxide; Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	Mylan Pharamceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Allura red AC dye	DIG Info	Solute carrier SLCO2B1 (Ki = 4.7 uM)	[2]
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Allura red AC dye	DIG Info	Solute carrier SLCO2B1 (Ki = 2.59 uM)	[5]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 3	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Sucralose; Mannitol; Butylated hydroxyanisole; Ferric oxide red; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Chewable Tablet
Company	Kremers Urban Pharmaceuticals Inc.
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sucralose	DIG Info	Carbonic anhydrase II (Ki = 300 nM)	[10]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Butylhydroxyanisole	DIG Info	Prostaglandin G/H synthase 2 (IC50 = 2.6 uM)	[2]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 4	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Sucralose; Mannitol; Butylated hydroxyanisole; Ferric oxide red; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Chewable Tablet
Company	AvKARE
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sucralose	DIG Info	Carbonic anhydrase II (Ki = 300 nM)	[10]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Butylhydroxyanisole	DIG Info	Prostaglandin G/H synthase 2 (IC50 = 2.6 uM)	[2]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 5	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Sucralose; Mannitol; Butylated hydroxyanisole; Ferric oxide red; Croscarmellose sodium; Silicon dioxide; Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	Proficient Rx
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sucralose	DIG Info	Carbonic anhydrase II (Ki = 300 nM)	[10]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Butylhydroxyanisole	DIG Info	Prostaglandin G/H synthase 2 (IC50 = 2.6 uM)	[2]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 6	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Sucralose; Mannitol; Butylated hydroxyanisole; Ferric oxide red; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Chewable Tablet
Company	AvPAK
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sucralose	DIG Info	Carbonic anhydrase II (Ki = 300 nM)	[10]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Butylhydroxyanisole	DIG Info	Prostaglandin G/H synthase 2 (IC50 = 2.6 uM)	[2]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 7	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium lauryl sulfate; Maltodextrin; Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Hydroxypropyl cellulose (type h); Sodium starch glycolate type a potato; Starch, corn
Dosage Form	Chewable Tablet
Company	Carilion Materials Management; Teva Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Dextrin	DIG Info	Colon cancer Caco-2 cells (Inhibition ratio > 55 %)	[8]
Drug Formulation 8	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium lauryl sulfate; Maltodextrin; Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Hydroxypropyl cellulose; Sodium starch glycolate type a potato; Starch, corn
Dosage Form	Chewable Tablet
Company	Physicians Total Care
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Dextrin	DIG Info	Colon cancer Caco-2 cells (Inhibition ratio > 55 %)	[8]
Drug Formulation 9	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium lauryl sulfate; Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Colloidal silicon dioxide; Hydroxypropyl cellulose (type el)
Dosage Form	Chewable Tablet
Company	Hangzhou Minsheng Binjiang Pharm
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 10	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Strawberry
Dosage Form	Chewable Tablet
Company	Jubilant Cadista Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 11	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Edetate disodium; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Macleods Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 12	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry
Dosage Form	Chewable Tablet
Company	A-S Medication Solutions; Torrent Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 13	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Dr Reddy's Laboratories
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 14	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Camber Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 15	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	A-S Medication Solutions; Par Pharmaceutical; Preferred Pharamaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 16	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Citron Pharma; Lucid Pharma
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 17	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cherry; Hydroxypropyl cellulose (type h); Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	Aurobindo Pharma
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 18	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose
Dosage Form	Chewable Tablet
Company	Bryant Ranch Prepack; Greenstone
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 19	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline
Dosage Form	Chewable Tablet
Company	American Health Packaging; Apotex
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 20	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	Ajanta Pharmaceutical
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 21	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Chewable Tablet
Company	ASE Direct; Bionpharma; Proficient Rx; Recipharm Pharmaservices; WellSpring Pharmaceutical
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 22	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose
Dosage Form	Chewable Tablet
Company	A-S Medication Solutions; Bryant Ranch Prepack; Dispensing Solution
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 23	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cherry; Hydroxypropyl cellulose (1200000 mw); Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	American Health Packaging
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 24	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cherry; Hydroxypropyl cellulose (1200000 mw); Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	Preferred Pharamaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 25	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry
Dosage Form	Chewable Tablet
Company	DirectRX
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 26	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cherry; Hydroxypropyl cellulose (1200000 mw); Microcrystalline cellulose
Dosage Form	Chewable Tablet
Company	Preferred Pharamaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 27	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sucralose; Magnesium stearate; Mannitol; Ferric oxide red; Cellulose, microcrystalline; Copovidone k25-31; Sodium starch glycolate type a potato
Dosage Form	Chewable Tablet
Company	West-Ward Pharmaceticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sucralose	DIG Info	Carbonic anhydrase II (Ki = 300 nM)	[10]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Montelukast 10 mg tablet			Click to Show/Hide the Full List of Formulation(s): 41 Formulation(s)
Drug Formulation 1	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium lauryl sulfate; Fd&c blue no. 2; Fd&c yellow no. 6; Magnesium stearate; Mannitol; Titanium dioxide; Triacetin; Croscarmellose sodium; Silicon dioxide; Hypromellose, unspecified; Microcrystalline cellulose; Polydextrose; Polyethylene glycol, unspecified
Dosage Form	Oral Tablet
Company	Cardinal Health; Mylan Pharamceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sunset yellow FCF	DIG Info	Solute carrier SLCO2B1 (Ki = 68.4 uM)	[5]
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	FD&C blue no. 2	DIG Info	Adenosine receptor A3 (IC50 = 1 uM)	[2]
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 2	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Mannitol; Talc; Titanium dioxide; Croscarmellose sodium; Polyvinyl alcohol; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose; Polyethylene glycols
Dosage Form	Oral Tablet
Company	Aphena Pharma Solutions-Tennessee
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Polyvinyl alcohol	DIG Info	Debrisoquine 4-hydroxylase (EC50 = 354.8 uM)	[12]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 3	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Mannitol; Talc; Titanium dioxide; Croscarmellose sodium; Polyvinyl alcohol; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Polyethylene glycols
Dosage Form	Oral Tablet
Company	AvPAK; Proficient Rx
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Polyvinyl alcohol	DIG Info	Debrisoquine 4-hydroxylase (EC50 = 354.8 uM)	[12]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 4	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Sodium lauryl sulfate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type e); Hypromellose 2910 (6 mpa.s); Starch, corn
Dosage Form	Oral Tablet
Company	Hangzhou Minsheng Binjiang Pharm
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 5	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Sodium stearyl fumarate; Mannitol; Talc; Titanium dioxide; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Polyethylene glycols; Polyvinyl alcohol, unspecified
Dosage Form	Oral Tablet
Company	Kremers Urban Pharmaceuticals Inc.
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Sodium stearyl fumarate	DIG Info	Leukemia K562 cells (IC50 = 20.2 ug.mL-1)	[11]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 6	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Aspartame; Magnesium stearate; Mannitol; Ferric oxide red; Croscarmellose sodium; Cellulose, microcrystalline; Cherry; Hydroxypropyl cellulose (type h)
Dosage Form	Oral Tablet
Company	Aphena Pharma Solutions-Tennessee
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Aspartame	DIG Info	Pregnane X receptor (Ki = 13 uM)	[2]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 7	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Isopropyl alcohol; Magnesium stearate; Edetate disodium; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromellose 2910 (6 mpa.s)
Dosage Form	Oral Tablet
Company	NuCare Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Isopropyl alcohol	DIG Info	Lymphoma P388/ADR cells (IC50 = 0.22 uM)	[13]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 8	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Isopropyl alcohol; Magnesium stearate; Edetate disodium; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromellose 2910 (6 mpa.s)
Dosage Form	Oral Tablet
Company	Macleods Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Isopropyl alcohol	DIG Info	Lymphoma P388/ADR cells (IC50 = 0.22 uM)	[13]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 9	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Mannitol; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose (type l); Hypromellose 2910 (6 mpa.s)
Dosage Form	Oral Tablet
Company	Contract Pharmacal; RemedyRepack; Unichem Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 10	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Mannitol; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose (1200000 mw); Hypromelloses
Dosage Form	Oral Tablet
Company	Legacy Pharmaceutical
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 11	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Mannitol; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose; Hypromelloses
Dosage Form	Oral Tablet
Company	Camber Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Mannitol	DIG Info	Glycine receptor alpha-1 (EC50 = 12589.25 nM)	[4]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 12	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Sodium lauryl sulfate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Hydroxypropyl cellulose (type h); Hypromellose 2910 (6 mpa.s); Sodium starch glycolate type a potato; Starch, corn
Dosage Form	Oral Tablet
Company	International Laboratories; Legacy Pharmaceutical; MedVantx; NCS HealthCare of KY, Inc dba Vangard Labs; Proficient Rx; RemedyRepack; Teva Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 13	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Sodium lauryl sulfate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Hydroxypropyl cellulose; Hypromellose 2910 (6 mpa.s); Sodium starch glycolate type a potato; Starch, corn
Dosage Form	Oral Tablet
Company	Physicians Total Care
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Sodium lauryl sulfate	DIG Info	Solute carrier SLCO2B1 (Ki = 1.98 uM)	[5]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 14	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Titanium dioxide; Croscarmellose sodium; Polyethylene glycol 400; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Oral Tablet
Company	Dr Reddy's Laboratories; RemedyRepack
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Polyethylene glycol 400	DIG Info	Albendazole monooxygenase (IC50 = 10.77 mg.mL-1)	[9]
Drug Formulation 15	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Titanium dioxide; Croscarmellose sodium; Polyethylene glycol 400; Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Microcrystalline cellulose
Dosage Form	Oral Tablet
Company	American Health Packaging
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Polyethylene glycol 400	DIG Info	Albendazole monooxygenase (IC50 = 10.77 mg.mL-1)	[9]
Drug Formulation 16	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Titanium dioxide; Croscarmellose sodium; Polyethylene glycol 400; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Oral Tablet
Company	Legacy Pharmaceutical
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Polyethylene glycol 400	DIG Info	Albendazole monooxygenase (IC50 = 10.77 mg.mL-1)	[9]
Drug Formulation 17	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Polyethylene glycol 3350; Polyvinyl alcohol; Cellulose, microcrystalline; Sodium starch glycolate type a potato
Dosage Form	Oral Tablet
Company	Avera McKennan Hospital; PD-Rx Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Polyvinyl alcohol	DIG Info	Debrisoquine 4-hydroxylase (EC50 = 354.8 uM)	[12]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Polyethylene glycol 3350	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 18	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Polyethylene glycol 3350; Polyvinyl alcohol; Cellulose, microcrystalline; Sodium starch glycolate type a potato
Dosage Form	Oral Tablet
Company	West-Ward Pharmaceticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Polyvinyl alcohol	DIG Info	Debrisoquine 4-hydroxylase (EC50 = 354.8 uM)	[12]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Polyethylene glycol 3350	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 19	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Anhydrous lactose; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Silicon dioxide; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromellose 2910 (5 mpa.s)
Dosage Form	Oral Tablet
Company	American Health Packaging; Apotex; Cardinal Health; Legacy Pharmaceutical
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Silicon dioxide	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
Drug Formulation 20	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Hypromellose; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose
Dosage Form	Oral Tablet
Company	Dispensing Solution
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Hypromellose	DIG Info	Cytochrome P450 3A5 (IC50 = 19.4 uM)	[12]
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 21	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Polyethylene glycol 6000; Hydroxypropyl cellulose (120000 mw); Hypromellose 2910 (6 mpa.s)
Dosage Form	Oral Tablet
Company	Preferred Pharamaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Polyethylene glycol 6000	DIG Info	Albendazole monooxygenase (Inhibition ratio < 70 %)	[9]
Drug Formulation 22	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Polyethylene glycol 6000; Hydroxypropyl cellulose (type l); Hypromellose 2910 (6 mpa.s)
Dosage Form	Oral Tablet
Company	Accord Healthcare; NuCare Pharmaceuticals; PD-Rx Pharmaceuticals; RemedyRepack
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Polyethylene glycol 6000	DIG Info	Albendazole monooxygenase (Inhibition ratio < 70 %)	[9]
Drug Formulation 23	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Polyethylene glycol 6000; Hydroxypropyl cellulose (type l); Hypromellose 2910 (6 mpa.s)
Dosage Form	Oral Tablet
Company	DirectRX; Proficient Rx
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
	Polyethylene glycol 6000	DIG Info	Albendazole monooxygenase (Inhibition ratio < 70 %)	[9]
Drug Formulation 24	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose, low substituted; Hypromelloses
Dosage Form	Oral Tablet
Company	Amneal Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 25	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Talc; Titanium dioxide; Polyethylene glycol 3350; Cellulose, microcrystalline; Polyvinyl alcohol, unspecified; Sodium starch glycolate type a potato
Dosage Form	Oral Tablet
Company	NCS HealthCare of KY, Inc dba Vangard Labs
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Polyethylene glycol 3350	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 26	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromellose 2910 (6 mpa.s)
Dosage Form	Oral Tablet
Company	Aurobindo Pharma; Citron Pharma; Lucid Pharma; State of Florida DOH Central Pharmacy
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 27	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Hydroxypropyl cellulose (type h); Hypromellose 2910 (6 mpa.s); Microcrystalline cellulose
Dosage Form	Oral Tablet
Company	Aurobindo Pharma
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 28	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose; Hypromellose 2910 (6 mpa.s)
Dosage Form	Oral Tablet
Company	Greenstone
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 29	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromellose 2910 (6 mpa.s)
Dosage Form	Oral Tablet
Company	A-S Medication Solutions; Torrent Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 30	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Oral Tablet
Company	Major Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 31	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose; Hypromelloses
Dosage Form	Oral Tablet
Company	Torrent Pharmaceuticals
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 32	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromellose 2910 (15000 mpa.s)
Dosage Form	Oral Tablet
Company	A-S Medication Solutions; Aidarex Pharmaceuticals; BluePoint Laboratories; Glenmark Pharmaceutials
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 33	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Oral Tablet
Company	Ajanta Pharmaceutical; Proficient Rx; RemedyRepack
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 34	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose; Hypromellose 2208 (15000 cps)
Dosage Form	Oral Tablet
Company	A-S Medication Solutions
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 35	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses; Polyethylene glycols
Dosage Form	Oral Tablet
Company	Sandoz
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 36	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromellose 2208 (100 mpa.s)
Dosage Form	Oral Tablet
Company	Cardinal Health; Carilion Materials Management; Major Pharmaceuticals; Par Pharmaceutical; Raritan Pharmaceuticals; RemedyRepack; State of Florida DOH Central Pharmacy
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 37	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hydroxypropyl cellulose; Hypromelloses; Polyethylene glycols
Dosage Form	Oral Tablet
Company	Bryant Ranch Prepack; Clinical Solutions Wholesale
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 38	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Hydroxypropyl cellulose (1200000 mw); Hypromellose, unspecified; Microcrystalline cellulose
Dosage Form	Oral Tablet
Company	Proficient Rx
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 39	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose (type h); Hypromelloses
Dosage Form	Oral Tablet
Company	ASE Direct; Bionpharma; Recipharm Pharmaservices; RemedyRepack; WellSpring Pharmaceutical
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 40	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose; Hypromelloses
Dosage Form	Oral Tablet
Company	Bryant Ranch Prepack
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]
Drug Formulation 41	DFM Info click to show the detail info of this DFM
All DIGs	Click to Show/Hide the Full List of DIGs in This DFM Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Titanium dioxide; Croscarmellose sodium; Carnauba wax; Cellulose, microcrystalline; Hydroxypropyl cellulose; Hypromelloses
Dosage Form	Oral Tablet
Company	Lake Eire Medical & Surgical Supply DBA Quality Care Products; Physicians Total Care
DIG(s) with Biological Activity
	DIG Name	DIG Info	Representative Biological Activity of This DIG	REF
	Magnesium stearate	DIG Info	Albendazole monooxygenase (Protein expression downregulation)	[7]
	Carmellose sodium	DIG Info	Albendazole monooxygenase (Protein expression upregulation)	[7]

References
1	FDA label for approved montelukast from the official website of the U.S. Food and Drug Administration.
2	The activities of drug inactive ingredients on biological targets. Science. 2020 Jul 24;369(6502):403-413.
3	O-alkylhydroxylamines as rationally-designed mechanism-based inhibitors of indoleamine 2,3-dioxygenase-1. Eur J Med Chem. 2016 Jan 27; 108:564-576.
4	Pharmacological property optimization for allosteric ligands: A medicinal chemistry perspective. Bioorg Med Chem Lett. 2017 Jun 1; 27(11):2239-2258.
5	Bacterial metabolism rescues the inhibition of intestinal drug absorption by food and drug additives. Proc Natl Acad Sci U S A. 2020 Jul 7;117(27):16009-16018.
6	Design, synthesis and biological studies of a library of NK1-Receptor Ligands Based on a 5-arylthiosubstituted 2-amino-4,6-diaryl-3-cyano-4H-pyran core: Switch from antagonist to agonist effect by chemical modification. Eur J Med Chem. 2017 Sep 29; 138:644-660.
7	Effects of commonly used excipients on the expression of CYP3A4 in colon and liver cells. Pharm Res. 2010 Aug;27(8):1703-12.
8	Interactions between human multidrug resistance related protein (MRP2; ABCC2) and excipients commonly used in self-emulsifying drug delivery systems (SEDDS). Int J Pharm. 2013 Apr 15;447(1-2):192-8.
9	Pharmaceutical excipients inhibit cytochrome P450 activity in cell free systems and after systemic administration. Eur J Pharm Biopharm. 2008 Sep;70(1):279-88.
10	Sweet Binders: Carbonic Anhydrase IX in Complex with Sucralose. ACS Med Chem Lett. 2018 May 10; 9(7):657-661.
11	Synthesis and evaluation of (-)-Massoialactone and analogues as potential anticancer and anti-inflammatory agents. Eur J Med Chem. 2014 Apr 9; 76:291-300.
12	Mediation of in vitro cytochrome p450 activity by common pharmaceutical excipients. Mol Pharm. 2013 Jul 1;10(7):2739-48.
13	Synthesis and evaluation of dihydropyrroloquinolines that selectively antagonize P-glycoprotein. J Med Chem. 2004 Mar 11; 47(6):1413-22.

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