Details of the Active Pharmaceutical Ingredient (API)
General Information of API (ID: D00725) | |||||
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Name |
Venlafaxine
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Synonyms |
Click to Show/Hide the Synonyms of This API
venlafaxine; 93413-69-5; Elafax; D,L-Venlafaxine; Venlafaxina; Venlafaxinum; Effexor; 1-(2-(dimethylamino)-1-(4-methoxyphenyl)ethyl)cyclohexanol; 1-[2-(Dimethylamino)-1-(4-methoxyphenyl)ethyl]cyclohexanol; 1-[2-(dimethylamino)-1-(4-methoxyphenyl)ethyl]cyclohexan-1-ol; Efectin; CHEBI:9943; Venlafaxine [INN:BAN]; NCGC00095109-01; Venlafaxinum [INN-Latin]; Venlafaxin; Venlafaxina [INN-Spanish]; Cyclohexanol, 1-[2-(dimethylamino)-1-(4-methoxyphenyl)ethyl]-; DSSTox_CID_3737; DSSTox_RID_77175; DSSTox_GSID_23737; Venlafexine; Efectin (TN); Venlafaxine (INN); CAS-93413-69-5; SR-01000762930; DL-Venlafaxine; Venflaxine EP; HSDB 6699; Spectrum_001671; SpecPlus_000842; Spectrum2_000542; Spectrum3_000989; Spectrum4_001115; Spectrum5_001516; CHEMBL637; EC 618-944-2; N,N,O-Didesmethylvenlafaxine; SCHEMBL35154; BSPBio_002657; KBioGR_001590; KBioSS_002151; MLS006011859; DivK1c_006938; SPECTRUM1504171; SPBio_000583; GTPL7321; DTXSID6023737; BDBM82071; KBio1_001882; KBio2_002151; KBio2_004719; KBio2_007287; KBio3_001877; HMS1922F05; HMS2090F04; HMS2093A12; HMS3714K11; HMS3886K14; Pharmakon1600-01504171; 1-{2-(dimethylamino)-1-[4-(methyloxy)phenyl]ethyl}cyclohexanol; HY-B0196; Tox21_111425; CCG-39577; MFCD00864385; N,N-dimethyl-2-(1-hydroxycyclohexyl)-2-(4-methoxyphenyl)ethylamine; NSC_62923; NSC758676; STK621394; AKOS005555049; Cyclohexanol, 1-(2-(dimethylamino)-1-(4-methoxyphenyl)ethyl)-, (+-)-; Tox21_111425_1; AC-1547; AT-6375; DB00285; MCULE-6632261838; NSC-758676; SDCCGSBI-0052740.P003; NCGC00095109-02; NCGC00095109-03; NCGC00095109-04; NCGC00095109-05; NCGC00095109-06; NCGC00095109-08; NCGC00095109-20; SMR002204138; WY-45655; SBI-0052740.P002; CAS_93413-69-5; CAS_99300-78-4; DB-057399; FT-0642242; FT-0675793; FT-0675795; C07187; D08670; AB00053751-08; AB00053751-10; AB00053751-11; AB00053751_12; AB00053751_13; 413V695; Q898407; SR-01000762930-3; SR-01000762930-4; BRD-A51714012-001-02-3; BRD-A51714012-003-01-1; 1-[2-dimethylamino-1-(4-methoxylphenyl)ethyl]cyclohexanol; (RS)-1-[2-(dimethylamino)-1-(4-methoxyphenyl)ethyl]cyclohexanol; 540726-98-5
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Clinical Status |
Approved
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Disease Indication | Major depressive disorder | ICD-11: 6A70 | [1] | ||
PubChem CID | |||||
Formula |
C17H27NO2
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Canonical SMILES |
CN(C)CC(C1=CC=C(C=C1)OC)C2(CCCCC2)O
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InChI |
1S/C17H27NO2/c1-18(2)13-16(17(19)11-5-4-6-12-17)14-7-9-15(20-3)10-8-14/h7-10,16,19H,4-6,11-13H2,1-3H3
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InChIKey |
PNVNVHUZROJLTJ-UHFFFAOYSA-N
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Click to Show/Hide the Molecular Data (Structure/Property) of This API | |||||
Structure |
<iframe style="width: 300px; height: 300px;" frameborder="0" src="https://embed.molview.org/v1/?mode=balls&cid=5656"></iframe>
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3D MOL | 2D MOL | ||||
Physicochemical Properties | Molecular Weight | 277.4 | Topological Polar Surface Area | 32.7 | |
XlogP | 2.9 | Complexity | 279 | ||
Heavy Atom Count | 20 | Rotatable Bond Count | 5 | ||
Hydrogen Bond Donor Count | 1 | Hydrogen Bond Acceptor Count | 3 | ||
Full List of Drug Formulations (DFMs) Containing This API | ||||||
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Venlafaxine 150 mg tablet | Click to Show/Hide the Full List of Formulation(s): 6 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; Fd&c red no. 40; Dibutyl sebacate; Magnesium stearate; Mannitol; Talc; Triethyl citrate; Crospovidone; Polyethylene glycol 3350; Polysorbate 20; Polysorbate 80; Polyvinyl alcohol; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Hypromellose 2208 (4000 cps); Methacrylic acid - ethyl acrylate copolymer (1:1) type a
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Polysorbate 20 | DIG Info | Cytochrome P450 2E1 (IC50 = 64.1 uM) | [5] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; Fd&c red no. 40; Dibutyl sebacate; Magnesium stearate; Mannitol; Talc; Triethyl citrate; Crospovidone; Polyethylene glycol 3350; Polysorbate 20; Polysorbate 80; Polyvinyl alcohol; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Hypromellose 2208 (4000 mpa.s); Methacrylic acid - ethyl acrylate copolymer (1:1) type a
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Polysorbate 20 | DIG Info | Cytochrome P450 2E1 (IC50 = 64.1 uM) | [5] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Povidone; Silicon dioxide; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Trigen Laboratories; Vertical Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose, unspecified form; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Silicon dioxide; Cellulose acetate; Hypromellose, unspecified; Microcrystalline cellulose; Polyethylene glycol, unspecified; Povidone, unspecified
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | UCB; Upstate Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Maltodextrin; Magnesium stearate; Talc; Titanium dioxide; Triacetin; Silicon dioxide; Ethylcellulose, unspecified; Hypromellose, unspecified; Microcrystalline cellulose; Polyethylene glycol, unspecified; Xanthan gum
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Golden State Medical Supply | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Dextrin | DIG Info | Colon cancer Caco-2 cells (Inhibition ratio > 55 %) | [10] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Maltodextrin; Magnesium stearate; Talc; Titanium dioxide; Triacetin; Silicon dioxide; Cellulose, microcrystalline; Ethylcelluloses; Hypromelloses; Polyethylene glycols; Xanthan gum
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Nostrum Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Dextrin | DIG Info | Colon cancer Caco-2 cells (Inhibition ratio > 55 %) | [10] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Venlafaxine 37.5 mg tablet | Click to Show/Hide the Full List of Formulation(s): 26 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; Fd&c red no. 40; Dibutyl sebacate; Magnesium stearate; Mannitol; Talc; Triethyl citrate; Crospovidone; Polyethylene glycol 3350; Polysorbate 20; Polysorbate 80; Polyvinyl alcohol; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Hypromellose 2208 (4000 cps); Methacrylic acid - ethyl acrylate copolymer (1:1) type a
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Polysorbate 20 | DIG Info | Cytochrome P450 2E1 (IC50 = 64.1 uM) | [5] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; Fd&c red no. 40; Dibutyl sebacate; Magnesium stearate; Mannitol; Talc; Triethyl citrate; Crospovidone; Polyethylene glycol 3350; Polysorbate 20; Polysorbate 80; Polyvinyl alcohol; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Hypromellose 2208 (4000 mpa.s); Methacrylic acid - ethyl acrylate copolymer (1:1) type a
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Polysorbate 20 | DIG Info | Cytochrome P450 2E1 (IC50 = 64.1 uM) | [5] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Povidone; Silicon dioxide; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Trigen Laboratories; Vertical Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Povidone; Silicon dioxide; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycol
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose, unspecified form; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Silicon dioxide; Cellulose acetate; Hypromellose, unspecified; Microcrystalline cellulose; Polyethylene glycol, unspecified; Povidone, unspecified
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | UCB; Upstate Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | DirectRX; Heritage Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols; Povidones
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Dosage Form | Oral Tablet | |||||
Company | A-S Medication Solutions; Aidarex Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; D&c yellow no. 10; Magnesium stearate; Cellulose, microcrystalline; Povidones; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Aphena Pharma Solutions-Tennessee; Clinical Solutions Wholesale; Qualitest Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Povidone; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | PD-Rx Pharmaceuticals; Stat Rx USA | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Crospovidone; Cellulose, microcrystalline
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Dosage Form | Oral Tablet | |||||
Company | Alembic Pharmaceuticals; NorthStar Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | A-S Medication Solutions; Aidarex Pharmaceuticals; NorthStar Rx; RemedyRepack; Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | TruPharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 15 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide yellow; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Aurobindo Pharma; Citron Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 16 |
DFM Info
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Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Teva Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 17 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Physicians Total Care; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 18 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Yaopharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 19 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 20 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Anhydrous lactose; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Aphena Pharma Solutions-Tennessee; AvKARE | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 21 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 22 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging; Cadila Healthcare; NCS HealthCare of KY, Inc dba Vangard Labs; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 23 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | BluePoint Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 24 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Colloidal silicon dioxide
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Dosage Form | Oral Tablet | |||||
Company | Rebel Distributors | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 25 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 26 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Colloidal silicon dioxide; Sodium starch glycolate type a potato; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Venlafaxine 75 mg tablet | Click to Show/Hide the Full List of Formulation(s): 26 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; Fd&c red no. 40; Dibutyl sebacate; Magnesium stearate; Mannitol; Talc; Triethyl citrate; Crospovidone; Polyethylene glycol 3350; Polysorbate 20; Polysorbate 80; Polyvinyl alcohol; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Hypromellose 2208 (4000 cps); Methacrylic acid - ethyl acrylate copolymer (1:1) type a
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Polysorbate 20 | DIG Info | Cytochrome P450 2E1 (IC50 = 64.1 uM) | [5] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; Fd&c red no. 40; Dibutyl sebacate; Magnesium stearate; Mannitol; Talc; Triethyl citrate; Crospovidone; Polyethylene glycol 3350; Polysorbate 20; Polysorbate 80; Polyvinyl alcohol; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Hypromellose 2208 (4000 mpa.s); Methacrylic acid - ethyl acrylate copolymer (1:1) type a
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products; RemedyRepack; Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Polysorbate 20 | DIG Info | Cytochrome P450 2E1 (IC50 = 64.1 uM) | [5] | |||
Polysorbate 80 | DIG Info | Prostaglandin G/H synthase 1 (IC50 = 1 uM) | [2] | |||
Polyvinyl alcohol | DIG Info | Debrisoquine 4-hydroxylase (EC50 = 354.8 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Polyethylene glycol 3350 | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Povidone; Silicon dioxide; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Trigen Laboratories; Vertical Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Povidone; Silicon dioxide; Cellulose acetate; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycol
|
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose, unspecified form; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Silicon dioxide; Cellulose acetate; Hypromellose, unspecified; Microcrystalline cellulose; Polyethylene glycol, unspecified; Povidone, unspecified
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | UCB; Upstate Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Contract Pharmacal; DirectRX; Heritage Pharmaceuticals; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols; Povidones
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Dosage Form | Oral Tablet | |||||
Company | Aidarex Pharmaceuticals; State of Florida DOH Central Pharmacy | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; D&c yellow no. 10; Magnesium stearate; Cellulose, microcrystalline; Povidones; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | A-S Medication Solutions; Aphena Pharma Solutions-Tennessee; Clinical Solutions Wholesale; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Qualitest Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Crospovidone; Cellulose, microcrystalline
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Dosage Form | Oral Tablet | |||||
Company | Alembic Pharmaceuticals; NorthStar Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | A-S Medication Solutions; Aidarex Pharmaceuticals; NorthStar Rx; PD-Rx Pharmaceuticals; RemedyRepack; Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | NuCare Pharmaceuticals; St Marys Medical Park Pharmacy; TruPharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide yellow; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Aurobindo Pharma; Citron Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 15 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Clinical Solutions Wholesale; RemedyRepack; Teva Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 16 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 17 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Yaopharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 18 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Anhydrous lactose; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Aphena Pharma Solutions-Tennessee; AvKARE | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 19 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 20 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | A-S Medication Solutions; American Health Packaging; Cadila Healthcare; Contract Pharmacal; H. J. Harkins Company; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Proficient Rx; Rebel Distributors; St Marys Medical Park Pharmacy; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 21 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | BluePoint Laboratories; Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 22 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Colloidal silicon dioxide
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Dosage Form | Oral Tablet | |||||
Company | Rebel Distributors | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 23 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 24 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Colloidal silicon dioxide; Sodium starch glycolate type a potato; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 25 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 26 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Crospovidone (15 mpa.s at 5%); Microcrystalline cellulose
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Dosage Form | Oral Tablet | |||||
Company | Clinical Solutions Wholesale; Proficient Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Venlafaxine 37.5 mg capsule | Click to Show/Hide the Full List of Formulation(s): 23 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Fd&c red no. 40; Butyl alcohol; Isopropyl alcohol; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Propylene glycol; Sodium hydroxide; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone; Alcohol; Ethylcellulose (100 mpa.s); Gelatin; Povidone k90; Shellac
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Orchid Chemicals & Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [7] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c red no. 28; Sodium lauryl sulfate; Fd&c blue no. 1; Fd&c yellow no. 6; Ferrosoferric oxide; Sodium bicarbonate; Talc; Titanium dioxide; Triethyl citrate; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Ethylcelluloses; Gelatin; Methacrylic acid - ethyl acrylate copolymer (1:1) type a
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Wockhardt | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
D&C red no. 28 | DIG Info | Organic anion transporter 1 (Ki = 0.064 uM) | [2] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c red no. 28; Sodium lauryl sulfate; Fd&c blue no. 1; Fd&c yellow no. 6; Ferrosoferric oxide; Sodium bicarbonate; Talc; Titanium dioxide; Triethyl citrate; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Ethylcelluloses; Gelatin; Methacrylic acid - ethyl acrylate copolymer (1:1) type a
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | American Health Packaging; Cardinal Health; Major Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
D&C red no. 28 | DIG Info | Organic anion transporter 1 (Ki = 0.064 uM) | [2] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c yellow no. 10; Dibutyl sebacate; Fd&c yellow no. 6; Ammonia; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin; Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Proficient Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium stearyl fumarate; Ammonia; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Talc; Titanium dioxide; Medium-chain triglycerides; Povidone; Cellulose, microcrystalline; Dimethylaminoethyl methacrylate - butyl methacrylate - methyl methacrylate copolymer; Ethylcelluloses; Gelatin; Shellac
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Dr Reddy's Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium stearyl fumarate | DIG Info | Leukemia K562 cells (IC50 = 20.2 ug.mL-1) | [9] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Medium-chain triglyceride | DIG Info | Colon cancer Caco-2 cells (Inhibition ratio > 36 %) | [10] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c yellow no. 10; Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin; Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | AvKARE; Clinical Solutions Wholesale; Lake Eire Medical & Surgical Supply DBA Quality Care Products; NCS HealthCare of KY, Inc dba Vangard Labs; Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c yellow no. 10; Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin, unspecified; Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | A-S Medication Solutions; Bryant Ranch Prepack; Teva Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c yellow no. 10; Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin; Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Fd&c blue no. 1; Talc; Titanium dioxide; Fd&c red no. 3; Ethylcelluloses; Gelatin; Hypromelloses; Polyethylene glycol
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Dosage Form | 24 HR Extended Release Capsule | |||||
Company | UDL Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
FD&C red no. 3 | DIG Info | Phosphodiesterase 3A (IC50 = 0.092 uM) | [2] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Silicon dioxide; Ethylcelluloses; Gelatin; Hypromelloses
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Torrent Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Silicon dioxide; Ethylcelluloses; Gelatin; Hypromelloses
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products; Major Pharmaceuticals; PD-Rx Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Cellulose, microcrystalline; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin; Hypromelloses
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Cadila Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Cellulose, microcrystalline; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin; Hypromelloses
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Golden State Medical Supply; Lake Eire Medical & Surgical Supply DBA Quality Care Products; NuCare Pharmaceuticals; RemedyRepack; TYA Pharmaceuticals; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin, unspecified; Hypromellose, unspecified; Microcrystalline cellulose
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Preferred Pharamaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 15 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Ethylcellulose (20 mpa.s); Gelatin; Hypromellose 2910 (5 mpa.s); Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Aphena Pharma Solutions-Tennessee; Aurobindo Pharma; Avera McKennan Hospital; Clinical Solutions Wholesale; Kaiser Foundation Hospitals; Lucid Pharma; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 16 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Ethylcellulose (20 mpa.s); Gelatin, unspecified; Hypromellose 2910 (5 mpa.s); Shellac; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 17 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Titanium dioxide; Cellulose, microcrystalline; Ethylcellulose, unspecified; Gelatin; Hydroxypropyl cellulose; Hypromelloses; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Macleods Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 18 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Carilion Materials Management | |||||
Drug Formulation 19 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin, unspecified; Hypromellose 2910 (6 mpa.s); Hypromellose, unspecified; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Greenstone | |||||
Drug Formulation 20 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Cardinal Health; Rebel Distributors | |||||
Drug Formulation 21 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Physicians Total Care | |||||
Drug Formulation 22 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin, unspecified; Hypromellose 2910 (6 mpa.s); Hypromellose, unspecified; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Pfizer | |||||
Drug Formulation 23 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Apotex; Medsource Pharmaceuticals; Proficient Rx; Rebel Distributors | |||||
Venlafaxine 75 mg capsule | Click to Show/Hide the Full List of Formulation(s): 25 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Fd&c red no. 40; Butyl alcohol; Isopropyl alcohol; Ferric oxide red; Ferric oxide yellow; Propylene glycol; Sodium hydroxide; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone; Alcohol; Ethylcellulose (100 mpa.s); Gelatin; Povidone k90; Shellac
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Orchid Chemicals & Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [7] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c yellow no. 10; Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Lecithin, soybean; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin; Shellac; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Proficient Rx; RxChange | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Soybean lecithin | DIG Info | Albendazole monooxygenase (IC50 = 6.61 mg.mL-1) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c red no. 28; Sodium lauryl sulfate; Fd&c blue no. 1; Fd&c yellow no. 6; Ferrosoferric oxide; Sodium bicarbonate; Talc; Titanium dioxide; Triethyl citrate; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Ethylcelluloses; Gelatin; Methacrylic acid - ethyl acrylate copolymer (1:1) type a
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Wockhardt | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
D&C red no. 28 | DIG Info | Organic anion transporter 1 (Ki = 0.064 uM) | [2] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c red no. 28; Sodium lauryl sulfate; Fd&c blue no. 1; Fd&c yellow no. 6; Ferrosoferric oxide; Sodium bicarbonate; Talc; Titanium dioxide; Triethyl citrate; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Ethylcelluloses; Gelatin; Methacrylic acid - ethyl acrylate copolymer (1:1) type a
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | American Health Packaging; Cardinal Health; Major Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
D&C red no. 28 | DIG Info | Organic anion transporter 1 (Ki = 0.064 uM) | [2] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c yellow no. 10; Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin; Shellac; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Aidarex Pharmaceuticals; AvKARE; Clinical Solutions Wholesale; Lake Eire Medical & Surgical Supply DBA Quality Care Products; MedVantx; NCS HealthCare of KY, Inc dba Vangard Labs; Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c yellow no. 10; Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin, unspecified; Shellac; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | A-S Medication Solutions; Bryant Ranch Prepack; Teva Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium stearyl fumarate; Ammonia; Ferric oxide red; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Talc; Titanium dioxide; Medium-chain triglycerides; Povidone; Cellulose, microcrystalline; Dimethylaminoethyl methacrylate - butyl methacrylate - methyl methacrylate copolymer; Ethylcelluloses; Gelatin; Shellac
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Dr Reddy's Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium stearyl fumarate | DIG Info | Leukemia K562 cells (IC50 = 20.2 ug.mL-1) | [9] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Medium-chain triglyceride | DIG Info | Colon cancer Caco-2 cells (Inhibition ratio > 36 %) | [10] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Fd&c blue no. 1; Fd&c yellow no. 5; Sucrose; Talc; Titanium dioxide; Silicon dioxide; Ethylcelluloses; Gelatin; Hypromelloses
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products; Major Pharmaceuticals; Preferred Pharamaceuticals; Torrent Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Hydrazine yellow | DIG Info | GABA(A) receptor alpha-1 (IC50 = 13 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c yellow no. 10; Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin; Shellac; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c red no. 28; Sodium lauryl sulfate; Fd&c blue no. 1; Talc; Titanium dioxide; Ethylcelluloses; Gelatin; Hypromelloses; Polyethylene glycol
|
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Dosage Form | 24 HR Extended Release Capsule | |||||
Company | UDL Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
D&C red no. 28 | DIG Info | Organic anion transporter 1 (Ki = 0.064 uM) | [2] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferric oxide red; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Cellulose, microcrystalline; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin; Hypromelloses
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | DirectRX | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferric oxide red; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Cellulose, microcrystalline; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin; Hypromelloses
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Cadila Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferric oxide red; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Cellulose, microcrystalline; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin; Hypromelloses
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Preferred Pharamaceuticals; RemedyRepack; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Cellulose, microcrystalline; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin; Hypromelloses
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Aphena Pharma Solutions-Tennessee; Golden State Medical Supply | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 15 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Ethylcellulose (20 mpa.s); Gelatin; Hypromellose 2910 (5 mpa.s); Shellac; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | A-S Medication Solutions; Aphena Pharma Solutions-Tennessee; Aurobindo Pharma; Avera McKennan Hospital; Clinical Solutions Wholesale; Kaiser Foundation Hospitals; Lucid Pharma; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 16 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Ethylcellulose (20 mpa.s); Gelatin, unspecified; Hypromellose 2910 (5 mpa.s); Shellac; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 17 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Ethylcellulose (20 mpa.s); Gelatin, unspecified; Hypromellose 2910 (5 mpa.s); Shellac; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 18 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Titanium dioxide; Cellulose, microcrystalline; Ethylcellulose, unspecified; Gelatin; Hydroxypropyl cellulose; Hypromelloses; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Macleods Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 19 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Carilion Materials Management | |||||
Drug Formulation 20 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin, unspecified; Hypromellose 2910 (6 mpa.s); Hypromellose, unspecified; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Greenstone | |||||
Drug Formulation 21 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Cardinal Health; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Rebel Distributors | |||||
Drug Formulation 22 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Apotex; DirectRX; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Medsource Pharmaceuticals; Physicians Total Care; Rebel Distributors; Unit Dose Services | |||||
Drug Formulation 23 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin, unspecified; Hypromellose 2910 (6 mpa.s); Hypromellose, unspecified; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | PD-Rx Pharmaceuticals; Pfizer; RemedyRepack | |||||
Drug Formulation 24 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | RemedyRepack | |||||
Drug Formulation 25 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | RemedyRepack | |||||
Venlafaxine 225 mg tablet | Click to Show/Hide the Full List of Formulation(s): 5 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Polyethylene glycol 1000; Povidone; Silicon dioxide; Cellulose, microcrystalline; Hypromelloses
|
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Clinical Solutions Wholesale | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 1000 | DIG Info | Cytochrome P450 2E1 (IC50 = 75.3 uM) | [5] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Povidone; Silicon dioxide; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
|
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Trigen Laboratories; Vertical Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose, unspecified form; Magnesium stearate; Mannitol; Ferrosoferric oxide; Propylene glycol; Titanium dioxide; Triacetin; Silicon dioxide; Cellulose acetate; Hypromellose, unspecified; Microcrystalline cellulose; Polyethylene glycol, unspecified; Povidone, unspecified
|
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | UCB; Upstate Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Mannitol | DIG Info | Glycine receptor alpha-1 (EC50 = 12589.25 nM) | [4] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Maltodextrin; Magnesium stearate; Talc; Titanium dioxide; Triacetin; Silicon dioxide; Ethylcellulose, unspecified; Hypromellose, unspecified; Microcrystalline cellulose; Polyethylene glycol, unspecified; Xanthan gum
|
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Golden State Medical Supply | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Dextrin | DIG Info | Colon cancer Caco-2 cells (Inhibition ratio > 55 %) | [10] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Maltodextrin; Magnesium stearate; Talc; Titanium dioxide; Triacetin; Silicon dioxide; Cellulose, microcrystalline; Ethylcelluloses; Hypromelloses; Polyethylene glycols; Xanthan gum
|
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Dosage Form | 24 HR Extended Release Oral Tablet | |||||
Company | Nostrum Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Dextrin | DIG Info | Colon cancer Caco-2 cells (Inhibition ratio > 55 %) | [10] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Venlafaxine 150 mg capsule | Click to Show/Hide the Full List of Formulation(s): 22 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c red no. 28; Sodium lauryl sulfate; Fd&c blue no. 1; Fd&c yellow no. 6; Ferrosoferric oxide; Sodium bicarbonate; Talc; Titanium dioxide; Triethyl citrate; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Ethylcelluloses; Gelatin; Methacrylic acid - ethyl acrylate copolymer (1:1) type a
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Wockhardt | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
D&C red no. 28 | DIG Info | Organic anion transporter 1 (Ki = 0.064 uM) | [2] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c red no. 28; Sodium lauryl sulfate; Fd&c blue no. 1; Fd&c yellow no. 6; Ferrosoferric oxide; Sodium bicarbonate; Talc; Titanium dioxide; Triethyl citrate; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Ethylcelluloses; Gelatin; Methacrylic acid - ethyl acrylate copolymer (1:1) type a
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | American Health Packaging; Cardinal Health; Major Pharmaceuticals; McKesson | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
FD&C blue no. 1 | DIG Info | Solute carrier SLCO2B1 (Ki = 13 uM) | [3] | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
D&C red no. 28 | DIG Info | Organic anion transporter 1 (Ki = 0.064 uM) | [2] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Butyl alcohol; Isopropyl alcohol; Ammonia; Ferric oxide red; Ferric oxide yellow; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Water; Polyethylene glycol 400; Alcohol; Ethylcellulose (100 mpa.s); Gelatin; Povidone k90; Shellac
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Orchid Chemicals & Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Isopropyl alcohol | DIG Info | Lymphoma P388/ADR cells (IC50 = 0.22 uM) | [7] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium stearyl fumarate; Ammonia; Ferric oxide red; Propylene glycol; Talc; Titanium dioxide; Medium-chain triglycerides; Povidone; Cellulose, microcrystalline; Dimethylaminoethyl methacrylate - butyl methacrylate - methyl methacrylate copolymer; Ethylcelluloses; Gelatin; Shellac
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Dr Reddy's Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium stearyl fumarate | DIG Info | Leukemia K562 cells (IC50 = 20.2 ug.mL-1) | [9] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Medium-chain triglyceride | DIG Info | Colon cancer Caco-2 cells (Inhibition ratio > 36 %) | [10] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Fd&c red no. 40; Fd&c yellow no. 5; Sucrose; Talc; Titanium dioxide; Silicon dioxide; Ethylcelluloses; Gelatin; Hypromelloses
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Lake Eire Medical & Surgical Supply DBA Quality Care Products; Major Pharmaceuticals; Torrent Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Hydrazine yellow | DIG Info | GABA(A) receptor alpha-1 (IC50 = 13 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
D&c red no. 28; Sodium lauryl sulfate; D&c yellow no. 10; Fd&c red no. 40; Talc; Titanium dioxide; Ethylcelluloses; Gelatin; Hypromelloses; Polyethylene glycol
|
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Dosage Form | 24 HR Extended Release Capsule | |||||
Company | UDL Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 4.7 uM) | [2] | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
D&C red no. 28 | DIG Info | Organic anion transporter 1 (Ki = 0.064 uM) | [2] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Allura red AC dye | DIG Info | Solute carrier SLCO2B1 (Ki = 2.59 uM) | [3] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Dibutyl sebacate; Fd&c yellow no. 6; Ammonia; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin, unspecified; Shellac; Starch, corn
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Proficient Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin; Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | A-S Medication Solutions; Aidarex Pharmaceuticals; AvKARE; Clinical Solutions Wholesale; Lake Eire Medical & Surgical Supply DBA Quality Care Products; McKesson; NCS HealthCare of KY, Inc dba Vangard Labs; Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Potassium hydroxide; Propylene glycol; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin, unspecified; Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | A-S Medication Solutions; Bryant Ranch Prepack; NuCare Pharmaceuticals; Teva Pharmaceuticals; Unit Dose Services | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Propylene glycol | DIG Info | Albendazole monooxygenase (Inhibition ratio < 20 %) | [8] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Dibutyl sebacate; Fd&c yellow no. 6; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Polyethylene glycol 400; Povidone k30; Ethylcellulose (7 mpa.s); Gelatin; Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Polyethylene glycol 400 | DIG Info | Albendazole monooxygenase (IC50 = 10.77 mg.mL-1) | [8] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferric oxide red; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Cellulose, microcrystalline; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin; Hypromelloses
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Cadila Healthcare | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferric oxide red; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Cellulose, microcrystalline; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin; Hypromelloses
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Aidarex Pharmaceuticals; Preferred Pharamaceuticals; RemedyRepack; TYA Pharmaceuticals; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Cetostearyl alcohol; Ferrosoferric oxide; Talc; Titanium dioxide; Silicon dioxide; Cellulose, microcrystalline; Ethyl acrylate and methyl methacrylate copolymer (2:1 750000 mw); Gelatin; Hypromelloses
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Aphena Pharma Solutions-Tennessee; Golden State Medical Supply | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Ethylcellulose (20 mpa.s); Gelatin; Hypromellose 2910 (5 mpa.s); Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Capsule | |||||
Company | Aurobindo Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 15 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Ethylcellulose (20 mpa.s); Gelatin; Hypromellose 2910 (5 mpa.s); Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Aphena Pharma Solutions-Tennessee; Aurobindo Pharma; Clinical Solutions Wholesale; Lucid Pharma; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 16 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferrosoferric oxide; Sucrose; Talc; Titanium dioxide; Ethylcellulose (20 mpa.s); Gelatin, unspecified; Hypromellose 2910 (5 mpa.s); Shellac; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 17 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Sodium lauryl sulfate; Ferric oxide red; Ferric oxide yellow; Ferrosoferric oxide; Titanium dioxide; Cellulose, microcrystalline; Ethylcellulose, unspecified; Gelatin; Hydroxypropyl cellulose; Hypromelloses; Starch, corn
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Macleods Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Drug Formulation 18 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin, unspecified; Hypromellose 2910 (6 mpa.s); Hypromellose, unspecified; Powdered cellulose
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Greenstone | |||||
Drug Formulation 19 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Aphena Pharma Solutions-Tennessee; Cardinal Health; Lake Eire Medical & Surgical Supply DBA Quality Care Products; Rebel Distributors | |||||
Drug Formulation 20 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Bryant Ranch Prepack; Physicians Total Care | |||||
Drug Formulation 21 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin, unspecified; Hypromellose 2910 (6 mpa.s); Hypromellose, unspecified; Powdered cellulose
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Pfizer; RemedyRepack | |||||
Drug Formulation 22 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ferric oxide red; Titanium dioxide; Ethylcellulose (100 mpa.s); Gelatin; Hypromellose 2910 (6 mpa.s); Hypromelloses; Powdered cellulose
|
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Dosage Form | 24 HR Extended Release Oral Capsule | |||||
Company | Apotex; Clinical Solutions Wholesale; DirectRX; Proficient Rx; Rebel Distributors | |||||
Venlafaxine 100 mg tablet | Click to Show/Hide the Full List of Formulation(s): 21 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | Heritage Pharmaceuticals; Kaiser Foundation Hospitals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; D&c yellow no. 10; Magnesium stearate; Cellulose, microcrystalline; Povidones; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Clinical Solutions Wholesale; Qualitest Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Povidone; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Kaiser Foundation Hospitals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Crospovidone; Cellulose, microcrystalline
|
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Dosage Form | Oral Tablet | |||||
Company | Aidarex Pharmaceuticals; Alembic Pharmaceuticals; NorthStar Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato; Starch, corn
|
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Dosage Form | Oral Tablet | |||||
Company | Avera McKennan Hospital; NorthStar Rx; Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | TruPharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide yellow; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Aurobindo Pharma; Citron Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Teva Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Physicians Total Care | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Yaopharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 15 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Anhydrous lactose; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | AvKARE | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 16 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 17 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Cadila Healthcare; Rebel Distributors; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 18 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | BluePoint Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 19 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Colloidal silicon dioxide
|
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Dosage Form | Oral Tablet | |||||
Company | Rebel Distributors | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 20 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 21 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Crospovidone (15 mpa.s at 5%)
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Dosage Form | Oral Tablet | |||||
Company | Proficient Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Venlafaxine 25 mg tablet | Click to Show/Hide the Full List of Formulation(s): 17 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | Heritage Pharmaceuticals; Kaiser Foundation Hospitals; RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; D&c yellow no. 10; Magnesium stearate; Cellulose, microcrystalline; Povidones; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Clinical Solutions Wholesale; Qualitest Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; D&c yellow no. 10; Magnesium stearate; Cellulose, microcrystalline; Povidone k12; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Povidone; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Kaiser Foundation Hospitals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Crospovidone; Cellulose, microcrystalline
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Dosage Form | Oral Tablet | |||||
Company | Aidarex Pharmaceuticals; Alembic Pharmaceuticals; NorthStar Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato; Starch, corn
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Dosage Form | Oral Tablet | |||||
Company | Avera McKennan Hospital; NorthStar Rx; RemedyRepack; Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | TruPharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide yellow; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Aurobindo Pharma; Citron Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Carilion Materials Management; RemedyRepack; Teva Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Yaopharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Anhydrous lactose; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | AvKARE | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 15 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging; Cadila Healthcare; Rebel Distributors; RemedyRepack; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 16 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | BluePoint Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 17 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Colloidal silicon dioxide
|
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Dosage Form | Oral Tablet | |||||
Company | Rebel Distributors | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Venlafaxine 50 mg tablet | Click to Show/Hide the Full List of Formulation(s): 17 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | RemedyRepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Povidone; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols
|
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Dosage Form | Oral Tablet | |||||
Company | DirectRX; Heritage Pharmaceuticals; Kaiser Foundation Hospitals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 3 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Titanium dioxide; Croscarmellose sodium; Cellulose, microcrystalline; Hypromelloses; Polyethylene glycols; Povidones
|
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Dosage Form | Oral Tablet | |||||
Company | Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Carmellose sodium | DIG Info | Albendazole monooxygenase (Protein expression upregulation) | [6] | |||
Drug Formulation 4 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Sodium lauryl sulfate; D&c yellow no. 10; Magnesium stearate; Cellulose, microcrystalline; Povidones; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Mylan Pharamceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Quinoline yellow WS | DIG Info | Estrogen receptor alpha (IC50 = 18 uM) | [2] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 5 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Fd&c yellow no. 6; Magnesium stearate; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
|||||
Dosage Form | Oral Tablet | |||||
Company | Clinical Solutions Wholesale; Qualitest Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sunset yellow FCF | DIG Info | Solute carrier SLCO2B1 (Ki = 68.4 uM) | [3] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 6 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Povidone; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
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Dosage Form | Oral Tablet | |||||
Company | Kaiser Foundation Hospitals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Povidone | DIG Info | Cholesterol 25-hydroxylase (IC50 = 78.3 uM) | [5] | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 7 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Crospovidone; Cellulose, microcrystalline
|
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Dosage Form | Oral Tablet | |||||
Company | Alembic Pharmaceuticals; NorthStar Rx | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Crospovidone | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 8 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato; Starch, corn
|
|||||
Dosage Form | Oral Tablet | |||||
Company | Aidarex Pharmaceuticals; NorthStar Rx; RemedyRepack; Sun Pharmaceutical Industries | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 9 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
|
|||||
Dosage Form | Oral Tablet | |||||
Company | TruPharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 10 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide yellow; Povidone k30; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Aurobindo Pharma; Citron Pharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 11 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Teva Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 12 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Silicon dioxide; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | Yaopharma | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Silicon dioxide | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 13 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Anhydrous lactose; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | AvKARE | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 14 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 15 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | American Health Packaging; Cadila Healthcare; RemedyRepack; Zydus Pharmaceuticals | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 16 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Microcrystalline cellulose; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | BluePoint Laboratories | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Drug Formulation 17 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Lactose monohydrate; Magnesium stearate; Ferric oxide red; Ferric oxide yellow; Cellulose, microcrystalline; Sodium starch glycolate type a potato
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Dosage Form | Oral Tablet | |||||
Company | NCS HealthCare of KY, Inc dba Vangard Labs | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
Venlafaxine Hydrochloride eq 37.5mg base extended release capsule | Click to Show/Hide the Full List of Formulation(s): 2 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Colloidal Silicon Dioxide; Cetostearyl Alcohol; Gelatin; Hypromellose; Microcrystalline Cellulose; Polyacrylate Dispersion; Sodium Lauryl Sulfate; Talc; Titanium Dioxide
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Dosage Form | Extended Release Capsule | |||||
Company | Bryant Ranch Prepack | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Sodium lauryl sulfate | DIG Info | Solute carrier SLCO2B1 (Ki = 1.98 uM) | [3] | |||
Gelatin | DIG Info | Mephenytoin 4-hydroxylase (EC50 = 20.5 uM) | [5] | |||
Hypromellose | DIG Info | Cytochrome P450 3A5 (IC50 = 19.4 uM) | [5] | |||
Drug Formulation 2 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Ethylcellulose; Hypromellose; Sugar Spheres
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Dosage Form | Extended Release Capsule | |||||
Company | Florida Pharmaceutical Products | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Hypromellose | DIG Info | Cytochrome P450 3A5 (IC50 = 19.4 uM) | [5] | |||
Venlafaxine Hydrochloride eq 12.5mg base tablet | Click to Show/Hide the Full List of Formulation(s): 1 Formulation(s) | |||||
Drug Formulation 1 |
DFM Info
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All DIGs | Click to Show/Hide the Full List of DIGs in This DFM
Cellulose; Iron Oxides; Lactose; Magnesium Stearate; Sodium Starch Glycolate
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Dosage Form | Tablet | |||||
Company | Wyeth Pharms | |||||
DIG(s) with Biological Activity | ||||||
DIG Name | DIG Info | Representative Biological Activity of This DIG | REF | |||
Magnesium stearate | DIG Info | Albendazole monooxygenase (Protein expression downregulation) | [6] | |||
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